SCHEMBL3932273

SCHEMBL3932273

[CH2]c1ccc(C(=O)N(CCC)c2ccncc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 3/20 0.44
PDE10A Q9Y233 2/20 0.42
NAMPT P43490 1/20 0.41
HTT P42858 1/20 0.40
ALDH1A1 P00352 2/20 0.39
ADRB2 P07550 1/20 0.39
KDM4E B2RXH2 1/20 0.39
KMT2A Q03164 1/20 0.39
EGFR P00533 1/20 0.38
ERBB2 P04626 1/20 0.38
MAPK14 Q16539 1/20 0.38
ACHE P22303 1/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
GRM1 Q13255 1/20 0.37
SLC6A2 P23975 1/20 0.37
ADRA2C P18825 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL95975 0.76 KDM4E (0.65) MLYCDPDE10ANAMPTHTTKDM4E
SCHEMBL27594794 0.74 SLC6A2 (0.42) MLYCDALDH1A1CA12CA9SLC6A2
SCHEMBL5543209 0.74 MLYCD (0.62) MLYCDALDH1A1EGFRERBB2TSHR
SCHEMBL18455023 0.73 EGFR (0.46) MLYCDALDH1A1ADRB2EGFRERBB2
SCHEMBL8016233 0.73 MLYCD (0.40) MLYCDALDH1A1KMT2AEGFRERBB2
SCHEMBL9001626 0.73 ADRA2C (0.65) MLYCDHTTALDH1A1ADRB2KMT2A
SCHEMBL2960979 0.72 USP2 (0.58) HTTALDH1A1KDM4EKMT2ATSHR
SCHEMBL8013240 0.71 ADRA2C (0.55) MLYCDPDE10AALDH1A1ADRB2ADRA2C
SCHEMBL1928093 0.71 PKM (0.54) MLYCDHTTALDH1A1ADRB2KMT2A
SCHEMBL9540613 0.71 MLYCD (0.57) MLYCDNAMPTALDH1A1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2043644-A1 NF- B INHIBITOR Otsuka Pharmaceutical Co., Ltd. (JP) 2009-04-08 EP disclosed
WO-2008010601-A1 NF- ϰB INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-01-24 WO disclosed