SCHEMBL3933302

SCHEMBL3933302

COC(=O)c1ccc(CCCCn2ccc([N+](=O)[O-])n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 2/20 0.50
CYP4F2 P78329 1/20 0.50
EP300 Q09472 7/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 2/20 0.45
POLB P06746 2/20 0.45
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
HRH1 P35367 1/20 0.41
FAAH O00519 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL185087 0.84 LMNA (0.53) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL3937034 0.81 EP300 (0.58) CYP4A11CYP4F2EP300SMN1; SMN2HRH1
SCHEMBL11118808 0.78 ALDH1A1 (0.51) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL27765548 0.77 POLB (0.46) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL1167139 0.74 KMT2A (0.51) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL1865448 0.74 ABHD6 (0.52) CYP4A11CYP4F2KMT2AMEN1ALDH1A1
SCHEMBL27787352 0.74 TDP1 (0.51) KMT2AALDH1A1POLBLMNASMN1; SMN2
SCHEMBL21961350 0.73 ALDH1A1 (0.44) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL29665356 0.73 LMNA (0.54) KMT2AMEN1ALDH1A1POLBLMNA
SCHEMBL31710511 0.73 KMT2A (0.49) KMT2AMEN1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2046755-A2 PYRAZOLES AS GLUCOKINASE ACTIVATORS F. Hoffmann-Roche AG (CH) 2009-04-15 EP disclosed
WO-2008012227-A2 PYRAZOLES AS GLUCOKINASE ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2008-01-31 WO disclosed