SCHEMBL3933847

SCHEMBL3933847

C[C@@H](Cc1cccc(CCNC(=O)OC(C)(C)C)c1)NC(=O)O

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.48
CTSK P43235 7/20 0.46
CTSS P25774 6/20 0.46
CTSB P07858 3/20 0.46
CTSL P07711 2/20 0.45
NQO2 P16083 1/20 0.45
POLB P06746 1/20 0.45
IDO1 P14902 1/20 0.44
SYK P43405 1/20 0.42
ATM Q13315 1/20 0.42
GLS O94925 1/20 0.42
NAMPT P43490 1/20 0.42
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5263829 0.88 CTSS (0.47) CTSKCTSSCTSBCTSLSYK
SCHEMBL693223 0.87 SIGMAR1 (0.53) CA2CTSKCTSSCTSBIDO1
SCHEMBL731698 0.85 CA2 (0.51) CA2CTSKCTSSCTSBCTSL
SCHEMBL6414451 0.85 CA2 (0.51) CA2CTSKCTSSCTSBCTSL
SCHEMBL731697 0.85 CA2 (0.51) CA2CTSKCTSSCTSBCTSL
SCHEMBL14977016 0.84 SIGMAR1 (0.50) CA2CTSKCTSSCTSBNQO2
SCHEMBL730856 0.84 SIGMAR1 (0.50) CA2CTSKCTSSCTSBNQO2
SCHEMBL730857 0.84 SIGMAR1 (0.50) CA2CTSKCTSSCTSBNQO2
SCHEMBL14987233 0.80 GLS (0.50) CA2CTSKNQO2POLBIDO1
SCHEMBL16798316 0.80 NQO2 (0.50) CA2CTSKNQO2POLBIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041118-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE Amgen, Inc (US) 2009-04-01 EP disclosed
WO-2007114827-A1 SUBSTITUTED HETEROCYCLIC COMPOUNDS AND METHODS OF USE AMGEN INC. (US) 2007-10-11 WO disclosed