SCHEMBL3936760

SCHEMBL3936760

COc1ccc(N)cc1C(=O)Nc1cccnc1

nearest known ligand 0.76

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.76
RAB9A P51151 3/20 0.68
MAPT P10636 2/20 0.68
NPC1 O15118 2/20 0.68
KDM4E B2RXH2 1/20 0.68
TSHR P16473 1/20 0.68
SMN1; SMN2 Q16637 1/20 0.68
LMNA P02545 1/20 0.64
POLB P06746 1/20 0.62
LRRK2 Q5S007 3/20 0.57
SGMS2 Q8NHU3 2/20 0.55
ALDH1A1 P00352 3/20 0.54
TP53 P04637 1/20 0.54
NAMPT P43490 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3934041 0.83 BRAF (0.63) MAPTNPC1KDM4EPOLBALDH1A1
SCHEMBL3934052 0.81 GAA (0.69) GAARAB9AMAPTNPC1KDM4E
SCHEMBL13162558 0.81 POLB (0.75) GAARAB9AMAPTNPC1KDM4E
SCHEMBL3487444 0.81 CYP11B2 (0.72) GAANPC1KDM4ESMN1; SMN2ALDH1A1
SCHEMBL3930125 0.81 CYP11B2 (0.68) KDM4ESMN1; SMN2ALDH1A1
SCHEMBL3940427 0.81 CYP11B2 (0.71) KDM4ELMNAALDH1A1TP53NAMPT
SCHEMBL4034779 0.80 GAA (0.53) GAARAB9AMAPTNPC1KDM4E
SCHEMBL2747860 0.80 LMNA (0.79) GAARAB9AMAPTNPC1KDM4E
SCHEMBL21022130 0.80 STAT3 (0.73) RAB9AMAPTNPC1SMN1; SMN2POLB
SCHEMBL12978039 0.79 GAA (0.84) GAARAB9AMAPTNPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831198-B1 PYRIDINE CARBOXAMIDE DERIVATIVES FOR USE AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2009-04-08 EP disclosed