SCHEMBL3939176

SCHEMBL3939176

COC(=O)c1[nH]c2c(-c3ccccc3)c(Cl)ccc2c(=O)c1Cc1ccc(C(=O)NC[C@@H]2CCCN2)cc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 7/20 0.40
MAPK8 P45983 5/20 0.39
MAPK9 P45984 4/20 0.39
CHUK O15111 1/20 0.39
CDK2 P24941 1/20 0.39
MAPK10 P53779 4/20 0.39
SUV39H2 Q9H5I1 2/20 0.38
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
DRD2 P14416 2/20 0.37
DRD3 P35462 2/20 0.37
SCN9A Q15858 1/20 0.37
PBK Q96KB5 1/20 0.37
PARP1 P09874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3940003 0.86 MAPK8 (0.52) MAPK8MAPK9MAPK10
SCHEMBL3634381 0.84 MAPK8 (0.53) MAPK8MAPK9MAPK10
SCHEMBL3634689 0.84 MAPK8 (0.42) MAPK8MAPK9MAPK10
SCHEMBL3631272 0.83 MAPK8 (0.44) MAPK8MAPK9MAPK10
SCHEMBL3938366 0.82 MAPK8 (0.52) MAPK8MAPK9MAPK10
SCHEMBL14604210 0.79 MAPK8 (0.51) MAPK8
SCHEMBL14604229 0.79 MAPK8 (0.49) MAPK8
SCHEMBL14604008 0.79 MAPK8 (0.48) MAPK8
SCHEMBL14604103 0.78 MAPK8 (0.51) MAPK8
SCHEMBL3635595 0.77 MAPK8 (0.40) MAPK8MAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009015917-A2 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. HOFFMANN-LA ROCHE AG (CH) 2009-02-05 WO disclosed