SCHEMBL3941624

SCHEMBL3941624

O=C(Nc1cccnc1Cl)c1cccc(C(F)(F)F)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.67
NNMT P40261 1/20 0.65
KCNQ3 O43525 2/20 0.62
KCNQ2 O43526 2/20 0.62
KCNE1 P15382 2/20 0.62
KCNQ1 P51787 2/20 0.62
KCNQ5 Q9NR82 1/20 0.62
GAA P10253 1/20 0.61
PTGS1 P23219 1/20 0.61
NPC1 O15118 2/20 0.59
RAB9A P51151 2/20 0.59
POLB P06746 2/20 0.59
TLR7 Q9NYK1 2/20 0.58
ALDH1A1 P00352 1/20 0.58
BRAF P15056 1/20 0.58
ALOX15 P16050 1/20 0.57
TSHR P16473 1/20 0.57
CASP1 P29466 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
HSD17B10 Q99714 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9868569 0.87 RAB9A (0.74) KMT2ANNMTKCNQ3KCNQ2KCNE1
SCHEMBL30733198 0.84 RAB9A (0.67) KMT2AGAAPTGS1NPC1RAB9A
SCHEMBL3933821 0.84 KCNQ3 (0.64) KMT2AKCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL28249147 0.84 RAB9A (0.67) KMT2AGAAPTGS1NPC1RAB9A
SCHEMBL14082710 0.83 RAB9A (0.58) KMT2ANNMTNPC1RAB9APOLB
SCHEMBL3941645 0.82 GAA (0.62) GAAPTGS1POLBTLR7ALDH1A1
SCHEMBL31606898 0.82 ALDH1A1 (0.62) GAAPTGS1TLR7ALDH1A1BRAF
SCHEMBL31606915 0.80 SCN5A (0.58) KMT2AKCNQ3KCNQ2KCNE1KCNQ1
SCHEMBL15492250 0.80 KMT2A (0.71) KMT2ANPC1RAB9APOLBALDH1A1
SCHEMBL4168687 0.79 CSF1R (0.72) KCNQ3KCNQ2KCNE1KCNQ1KCNQ5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831198-B1 PYRIDINE CARBOXAMIDE DERIVATIVES FOR USE AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2009-04-08 EP disclosed