SCHEMBL3941645

SCHEMBL3941645

COc1ncccc1NC(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.62
PTGS1 P23219 1/20 0.58
SCN5A Q14524 1/20 0.58
SCN9A Q15858 1/20 0.58
POLB P06746 1/20 0.57
P2RY1 P47900 2/20 0.57
BRAF P15056 5/20 0.56
TRPV1 Q8NER1 1/20 0.56
ALDH1A1 P00352 1/20 0.56
ALOX15 P16050 1/20 0.55
TSHR P16473 1/20 0.55
CASP1 P29466 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
HSD17B10 Q99714 1/20 0.55
RXFP1 Q9HBX9 2/20 0.54
CSF1R P07333 1/20 0.54
TLR7 Q9NYK1 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3941624 0.82 KMT2A (0.67) GAAPTGS1POLBBRAFTRPV1
SCHEMBL28249147 0.81 RAB9A (0.67) GAAPTGS1BRAFALDH1A1NPSR1
SCHEMBL30733198 0.81 RAB9A (0.67) GAAPTGS1BRAFALDH1A1NPSR1
SCHEMBL31282022 0.81 MEN1 (0.49) SCN5ASCN9APOLBTRPV1
SCHEMBL31606898 0.81 ALDH1A1 (0.62) GAAPTGS1SCN5ASCN9ABRAF
SCHEMBL26623448 0.78 POLB (0.60) POLBALDH1A1HSD17B10CYP1A2CYP3A4
SCHEMBL26623509 0.77 HDAC1 (0.51) GAASCN5ASCN9APOLB
SCHEMBL29572307 0.77 SORT1 (0.65) GAAPTGS1POLBBRAFTRPV1
SCHEMBL24274892 0.77 KCNQ3 (0.61) GAAPTGS1BRAFCSF1R
SCHEMBL21870341 0.77 GAA (1.00) GAAPTGS1POLBBRAFALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831198-B1 PYRIDINE CARBOXAMIDE DERIVATIVES FOR USE AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2009-04-08 EP disclosed