Prednicarbate

Prednicarbate

SCHEMBL3942

CCOC(=O)O[C@@]1(C(=O)COC(=O)CC)CC[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@H]3[C@H](O)C[C@@]21C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1

The experimentally established mechanism targets of Prednicarbate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 10/20 1.00
PGR P06401 8/20 1.00
HIF1A Q16665 5/20 1.00
LMNA P02545 3/20 1.00
CYP3A4 P08684 2/20 1.00
USP2 O75604 1/20 1.00
CYP2D6 P10635 1/20 1.00
CYP2C9 P11712 1/20 1.00
ABCB11 O95342 2/20 0.75
NR1I2 O75469 2/20 0.75
ABCC3 O15438 1/20 0.75
AR P10275 2/20 0.60
CHRM1 P11229 1/20 0.60
NR3C2 P08235 3/20 0.57
HSD17B10 Q99714 2/20 0.57
TNF P01375 1/20 0.57
IL6 P05231 1/20 0.57
SERPINA6 P08185 1/20 0.57
GLUL P15104 1/20 0.57
ADAM17 P78536 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prednicarbate SCHEMBL3941 1.00 NR3C1 (1.00) NR3C1PGRHIF1ALMNACYP3A4
Prednicarbate SCHEMBL5483489 1.00 NR3C1 (1.00) NR3C1PGRHIF1ALMNACYP3A4
Prednicarbate SCHEMBL1650745 1.00 NR3C1 (1.00) NR3C1PGRHIF1ALMNACYP3A4
Prednicarbate SCHEMBL6466947 0.98 NR3C1 (0.97) NR3C1PGRHIF1ALMNACYP3A4
Prednicarbate SCHEMBL30697296 0.95 NR3C1 (0.91) NR3C1PGRHIF1ALMNACYP3A4
SCHEMBL11430405 0.95 NR3C1 (0.90) NR3C1PGRHIF1ALMNACYP3A4
SCHEMBL11425522 0.94 NR3C1 (0.89) NR3C1PGRHIF1ALMNACYP3A4
SCHEMBL423275 0.94 NR3C1 (0.89) NR3C1PGRHIF1ALMNACYP3A4
SCHEMBL11431033 0.94 NR3C1 (0.88) NR3C1PGRHIF1ALMNACYP3A4
SCHEMBL20365864 0.94 PGR (0.88) NR3C1PGRHIF1ALMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12909 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137657-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
US-20260137656-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-20260034056-A1 PHARMACEUTICAL COMPOSITIONS FOR TREATING OCULAR DISEASES OR DISORDERS ALCON INC (CH) 2026-02-05 US claimed
US-20260027255-A1 Cross-Linked Telechelic Polymer Compositions, Methods of Preparation Thereof, and Methods of Using Same BETTY YU SKIN TECH ADVISORS LLC (US) 2026-01-29 US claimed
EP-4683679-A1 METHOD FOR DIAGNOSING AND TREATING NIS-EXPRESSING CARCINOMAS AND METASTASES NUSKE, Andreas (DE) 2026-01-28 EP claimed
EP-4301343-B1 PHARMACEUTICAL COMPOSITIONS WITH REDUCED SIDE EFFECT AND METHODS OF USING THE SAME TLC BIOPHARMACEUTICALS INC (US) 2025-11-19 EP claimed
US-20250319104-A1 MOISTURIZING CREAM FOR RADIATION DERMATITIS PERRY ARTHUR W (US) 2025-10-16 US claimed
US-20250312274-A1 A PHARMACEUTICAL FORMULATION FOR PRESSURISED METERED DOSE INHALER CHIESI FARMACEUTICI S.P.A. (IT) 2025-10-09 US claimed
EP-0900233-A1 NOVEL STEROID NITRITE AND NITRATE ESTER DERIVATIVES USEFUL AS ANTI-INFLAMMATORY DRUGS G.D. SEARLE & CO. (US) 1999-03-10 EP claimed
CN-1209318-A Nailpolish having function of resisting psoriasis HOECHST MARION ROUSSEL DE GMBH (DE) 1999-03-03 CN claimed
US-5858410-A Pharmaceutical nanosuspensions for medicament administration as systems with increased saturation solubility and rate of solution MEDAC GESELLSCHAFT FUR KLINISCHE SPEZIALPRAPARATE (DE) 1999-01-12 US claimed
WO-1997041144-A1 NOVEL STEROID NITRITE AND NITRATE ESTER DERIVATIVES USEFUL AS ANTI-INFLAMMATORY DRUGS G.D. SEARLE & CO. (US) 1997-11-06 WO claimed
WO-1997027862-A1 SUPPLEMENTATION OF GLUCOCORTICOIDS BELLARA MEDICAL PRODUCTS LIMITED (AU) 1997-08-07 WO claimed
WO-1997015298-A1 COMBINATION OF LTD, RECEPTOR ANTAGONISTS WITH GLUCOCORTICOSTEROIDS BAYER AKTIENGESELLSCHAFT (DE) 1997-05-01 WO claimed
EP-0675722-A1 HYDROXY VITAMIN D3 COMPOUNDS FOR TREATING SKIN ATROPHY LEO PHARMACEUTICAL PRODUCTS LTD. A/S (LOVENS KEMISKE FABRIK PRODUKTIONSAKTIESELSKAB) (DK) 1995-10-11 EP claimed
US-5407663-A Swishing solution in mouth, expectorating EISEN DRORE (US) 1995-04-18 US claimed
WO-1994014453-A1 HYDROXY VITAMIN D3 COMPOUNDS FOR TREATING SKIN ATROPHY Leo Pharmaceutical Products Ltd. A/S (Løvens Kemiske Fabrik Produktionsaktieselskab) (DK) 1994-07-07 WO claimed
EP-0496520-A1 Novel bone acting agents MERCK & CO. INC. (US) 1992-07-29 EP claimed