SCHEMBL3942876

SCHEMBL3942876

CCCN(C1CCN(CCN)CC1)S(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.51
HTR2C P28335 6/20 0.51
ALDH1A1 P00352 3/20 0.51
GAA P10253 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
CACNA1B Q00975 1/20 0.48
CACNA1C Q13936 1/20 0.48
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
TSHR P16473 3/20 0.44
HTT P42858 1/20 0.44
ATM Q13315 1/20 0.44
DRD2 P14416 1/20 0.43
HTR7 P34969 4/20 0.43
MMP3 P08254 3/20 0.42
CCR5 P51681 1/20 0.42
RORC P51449 1/20 0.42
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3568841 0.91 HTR2A (0.53) HTR2AHTR2CALDH1A1GAAL3MBTL1
SCHEMBL3556337 0.86 HTR2A (0.49) HTR2AHTR2CALDH1A1GAACACNA1B
SCHEMBL3556156 0.79 SLC6A2 (0.58) HTR2AHTR2CALDH1A1GAAL3MBTL1
SCHEMBL4017004 0.77 HTR2A (0.51) HTR2AHTR2CALDH1A1GAATSHR
SCHEMBL3941201 0.77 TSHR (0.48) HTR2AHTR2CALDH1A1GAAL3MBTL1
SCHEMBL19558635 0.76 ALDH1A1 (0.49) HTR2AHTR2CALDH1A1GAAL3MBTL1
SCHEMBL3556782 0.76 RXFP1 (0.43) CACNA1BCACNA1CMEN1LMNAMAPT
SCHEMBL3564132 0.73 RXFP1 (0.42) CACNA1BCACNA1CMEN1LMNAKMT2A
SCHEMBL3559225 0.71 DRD2 (0.47) HTR2AHTR2CALDH1A1GAAL3MBTL1
SCHEMBL14045161 0.71 HTR1A (0.40) HTR2AHTR2CALDH1A1GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1670470-B1 PYRIDINE DERIVATIVES AND USE THEREOF AS UROTENSIN II ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2009-04-08 EP disclosed