SCHEMBL3944253

SCHEMBL3944253

N#Cc1cccc(C(=CC=CC(=O)O)c2ccc(Cl)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 1/20 0.42
GSK3B P49841 2/20 0.42
S1PR1 P21453 1/20 0.41
S1PR3 Q99500 1/20 0.41
CNR1 P21554 2/20 0.39
ESR1 P03372 1/20 0.39
CNR2 P34972 1/20 0.39
P4HB P07237 6/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
GRM5 P41594 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
P2RX1 P51575 1/20 0.37
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3944250 1.00 VNN1 (0.42) VNN1GSK3BS1PR1S1PR3CNR1
SCHEMBL3944317 0.88 GSK3B (0.42) GSK3BESR1P4HBGRM5CES2
SCHEMBL3944310 0.88 GSK3B (0.42) GSK3BESR1P4HBGRM5CES2
SCHEMBL3944308 0.88 GSK3B (0.42) GSK3BESR1P4HBGRM5CES2
SCHEMBL3946828 0.84 P4HB (0.41) VNN1GSK3BESR1P4HBMAOB
SCHEMBL3946826 0.84 P4HB (0.41) VNN1GSK3BESR1P4HBMAOB
SCHEMBL3940491 0.84 NR1H4 (0.44) VNN1GSK3BESR1P4HB
SCHEMBL3946830 0.84 P4HB (0.41) VNN1GSK3BESR1P4HBMAOB
SCHEMBL3940487 0.84 NR1H4 (0.44) VNN1GSK3BESR1P4HB
SCHEMBL4098216 0.82 CES2 (0.53) MAOBL3MBTL1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090203667-A1 PENTADIENAMIDE DERIVATIVES KYOWA HAKKO KIRIN CO., LTD. (JP) 2009-08-13 US disclosed
EP-2050734-A1 PENTADIENAMIDE DERIVATIVE Kyowa Hakko Kirin Co., Ltd. (JP) 2009-04-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090203667-A1 PENTADIENAMIDE DERIVATIVES PRMT1, REN, NGLY1 VNN1 1184/4885GSK3B 3499/4885S1PR1 3100/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.