SCHEMBL3944871

SCHEMBL3944871

O=C1NC(CCc2ccccc2Cl)=C(C(=O)OCc2ccccc2)C(c2ccccn2)N1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.44
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 2/20 0.42
ADORA2B P29275 3/20 0.41
TP53 P04637 1/20 0.41
KDM4E B2RXH2 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3947142 0.86 MEN1 (0.53) MEN1KMT2AALDH1A1TP53KDM4E
SCHEMBL13942611 0.86 MEN1 (0.51) MEN1KMT2AALDH1A1TP53KDM4E
SCHEMBL3950394 0.85 MEN1 (0.56) HTTMEN1KMT2AALDH1A1TP53
SCHEMBL3944408 0.83 TSHR (0.49) HTTADORA2BTP53
SCHEMBL3951091 0.83 HTT (0.43) HTTMEN1KMT2ATP53KDM4E
SCHEMBL13942605 0.82 TSHR (0.52) HTTMEN1KMT2AALDH1A1TP53
SCHEMBL3944971 0.81 MEN1 (0.48) HTTMEN1KMT2AALDH1A1TP53
SCHEMBL3943138 0.81 RXFP1 (0.55) MEN1KMT2AALDH1A1
SCHEMBL13942363 0.81 ADORA2B (0.55) MEN1KMT2AADORA2B
SCHEMBL13942609 0.80 PKM (0.52) MEN1KMT2AALDH1A1TP53KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009020457-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-02-12 WO disclosed
WO-2009020457-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-02-12 WO disclosed