SCHEMBL3948717

SCHEMBL3948717

COc1ccc(Cl)cc1S(=O)(=O)N[C@@H]1C[C@H](CNC(=O)Oc2ccccc2)[N+](C(=O)[O-])(C(C)(C)C)C1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CPT1A P50416 2/20 0.46
CPT1B Q92523 2/20 0.46
CPT2 P23786 1/20 0.46
DRD2 P14416 4/20 0.39
ADRA1D P25100 4/20 0.39
ADRA1A P35348 4/20 0.39
ADRA1B P35368 4/20 0.39
KMT2A Q03164 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
GAA P10253 1/20 0.37
USP2 O75604 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TSHR P16473 2/20 0.37
NPC1 O15118 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
TP53 P04637 1/20 0.36
CASP1 P29466 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3951883 0.84 L3MBTL1 (0.44) CPT1ACPT1BCPT2DRD2ADRA1D
SCHEMBL3949063 0.80 L3MBTL1 (0.47) CPT1ACPT1BCPT2DRD2ADRA1D
SCHEMBL3950301 0.78 CPT2 (0.41) CPT1ACPT1BCPT2DRD2ADRA1D
SCHEMBL13662066 0.78 CPT1A (0.54) CPT1ACPT1BCPT2DRD2ADRA1D
SCHEMBL4294665 0.77 CPT2 (0.53) CPT1ACPT1BCPT2DRD2ADRA1D
SCHEMBL3947805 0.76 CTSL (0.47) KMT2AL3MBTL1SMN1; SMN2TP53CASP1
SCHEMBL8045577 0.75 CPT2 (0.50) CPT1ACPT1BCPT2DRD2ADRA1D
SCHEMBL3952237 0.74 L3MBTL1 (0.45) DRD2ADRA1DADRA1AADRA1BKMT2A
SCHEMBL3954902 0.73 KMT2A (0.47) DRD2ADRA1DADRA1AADRA1BKMT2A
SCHEMBL3950238 0.73 MAPK1 (0.37) KMT2AGAASMN1; SMN2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026197-A1 NOVEL CATHEPSIN C INHIBITORS AND THEIR USE GLAXO GROUP LIMITED (GB) 2009-02-26 WO disclosed