SCHEMBL3955073

SCHEMBL3955073

CCCCc1nc2ccc(F)cn2c(=O)c1-c1ccc(NC2CCN(C(=O)O)C2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
GFER P55789 4/20 0.35
ATM Q13315 1/20 0.35
RCE1 Q9Y256 1/20 0.35
HPGD P15428 1/20 0.34
CCNK O75909 2/20 0.34
CCNA2 P20248 2/20 0.34
CDK2 P24941 2/20 0.34
CDK7 P50613 2/20 0.34
CCNH P51946 2/20 0.34
MNAT1 P51948 2/20 0.34
CDK12 Q9NYV4 2/20 0.34
MCHR1 Q99705 1/20 0.34
MLNR O43193 1/20 0.34
USP30 Q70CQ3 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3962925 0.91 KDM4E (0.36) KDM4EALDH1A1GFERATMHPGD
SCHEMBL5131458 0.89 MET (0.44) ENPP2ALDH1A1MAPTUSP30
SCHEMBL5132205 0.89 MET (0.44) ENPP2ALDH1A1MAPTUSP30
SCHEMBL3961800 0.87 AGTR1 (0.43) KDM4EALDH1A1GAAMAPTGFER
SCHEMBL3963648 0.83 RHOC (0.35) GFERMCHR1MLNRKMT2A
SCHEMBL3955475 0.82 AXL (0.37) ENPP2
SCHEMBL3955467 0.82 AXL (0.37) ENPP2
SCHEMBL3961045 0.82 GFER (0.49) MAPTGFERKMT2A
Hydrochloric Acid SCHEMBL5128628 0.82 AXL (0.36) ENPP2
SCHEMBL3963579 0.82 AGTR1 (0.44) KDM4EALDH1A1GAAMAPTGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079737-A1 PYRIDOPYRIMIDINONE COMPOUNDS USEFUL IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2009-07-22 EP claimed
WO-2008097991-A1 PYRIDOPYRIMIDINONE COMPOUNDS USEFUL IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-08-14 WO claimed
EP-2079737-A1 PYRIDOPYRIMIDINONE COMPOUNDS USEFUL IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2009-07-22 EP disclosed
WO-2008097991-A1 PYRIDOPYRIMIDINONE COMPOUNDS USEFUL IN TREATING SODIUM CHANNEL-MEDIATED DISEASES OR CONDITIONS XENON PHARMACEUTICALS INC. (CA) 2008-08-14 WO disclosed