SCHEMBL3957451

SCHEMBL3957451

[CH2]CCN1CCN(CCC2CCOCC2)CC1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
DRD2 P14416 13/20 0.34
HTR2A P28223 13/20 0.34
DRD3 P35462 13/20 0.34
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3950050 0.89 ALDH1A1 (0.38) ALDH1A1KDM4EDRD2HTR2ADRD3
SCHEMBL3952872 0.89 PIM1 (0.30)
SCHEMBL3951154 0.82 DRD2 (0.37) ALDH1A1KDM4EDRD2HTR2ADRD3
SCHEMBL3950179 0.82 DRD2 (0.35) ALDH1A1KDM4EDRD2HTR2ADRD3
SCHEMBL12397 0.82 CYP1A2 (0.42) ALDH1A1KDM4EDRD2HTR2ADRD3
SCHEMBL12120559 0.81 ALOX15 (0.50) ALDH1A1KDM4EDRD2HTR2ADRD3
SCHEMBL13062 0.80 CYP1A2 (0.46) ALDH1A1CYP1A2
SCHEMBL3954983 0.79 KEAP1 (0.32) ALDH1A1
SCHEMBL3951360 0.78 ALDH1A1 (0.38) ALDH1A1KDM4EDRD2DRD3CYP1A2
SCHEMBL8233850 0.77 ALDH1A1 (0.46) ALDH1A1KDM4EDRD2DRD3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009024825-A1 2-PYRAZINYLBENZIMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-02-26 WO disclosed