SCHEMBL3961796

SCHEMBL3961796

Cc1nc2ccc(Br)cc2c(-c2ccc(F)cc2)c1CCO

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 3/20 0.48
PRNP P04156 1/20 0.48
PPARG P37231 1/20 0.48
NR2E3 Q9Y5X4 1/20 0.48
NCOR2 Q9Y618 1/20 0.48
ALDH1A1 P00352 2/20 0.47
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
CASP3 P42574 4/20 0.43
DPP4 P27487 1/20 0.41
KDM4E B2RXH2 1/20 0.40
DHODH Q02127 2/20 0.40
AURKA O14965 2/20 0.40
AURKB Q96GD4 2/20 0.40
KDR P35968 1/20 0.40
HTT P42858 2/20 0.40
AKR1B10 O60218 1/20 0.39
PTGFR P43088 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3970472 0.82 RXFP1 (0.47) RXFP1PRNPPPARGNR2E3NCOR2
SCHEMBL3969545 0.80 RXFP1 (0.45) RXFP1PRNPPPARGNR2E3NCOR2
SCHEMBL3962968 0.79 IDO1 (0.42) ALDH1A1DPP4KDM4ELMNAPRKAA2
SCHEMBL3970478 0.78 KDM4E (0.47) ALDH1A1KDM4E
SCHEMBL13881531 0.78 RXFP1 (0.60) RXFP1PRNPPPARGNR2E3NCOR2
SCHEMBL3970605 0.78 PRNP (0.79) RXFP1PRNPPPARGNR2E3NCOR2
SCHEMBL3970468 0.77 ALDH1A1 (0.79) RXFP1PRNPPPARGNR2E3NCOR2
SCHEMBL13881528 0.77 ALDH1A1 (0.60) RXFP1PRNPPPARGNR2E3NCOR2
SCHEMBL3961795 0.77 RXFP1 (0.49) RXFP1PRNPPPARGNR2E3NCOR2
SCHEMBL13881529 0.76 RXFP1 (0.48) RXFP1PRNPPPARGNR2E3NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009041904-A1 QUINOLINE COMPOUNDS HAVING AN ACTIVITY AGAINST THE GABAB RECEPTOR ASTRAZENECA AB (SE) 2009-04-02 WO disclosed