SCHEMBL3962368

SCHEMBL3962368

COC(=O)c1ccc(-c2cc(NCC3CC3)ncn2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR39 O43194 1/20 0.51
CLK4 Q9HAZ1 6/20 0.47
CYP1A2 P05177 6/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2D6 P10635 2/20 0.47
USP2 O75604 1/20 0.47
ALDH1A1 P00352 5/20 0.47
HSD17B10 Q99714 4/20 0.47
ALOX15 P16050 2/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HRH4 Q9H3N8 1/20 0.44
FAAH O00519 3/20 0.44
ADORA3 P0DMS8 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ROCK2 O75116 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2585526 0.77 ACACB (0.51) GPR39CLK4CYP1A2CYP3A4CYP2D6
SCHEMBL2584992 0.76 GPR39 (0.56) GPR39CLK4CYP1A2CYP3A4CYP2D6
SCHEMBL25836238 0.76 MAPK1 (0.50) MEN1KMT2AKDM4EPIM1
SCHEMBL17634546 0.74 PDE10A (0.43) GPR39CLK4CYP1A2CYP3A4CYP2D6
SCHEMBL19355384 0.73 PDE10A (0.44) GPR39CLK4CYP1A2CYP3A4CYP2D6
SCHEMBL2774028 0.73 S1PR1 (0.61) GPR39MEN1KMT2AHRH4KDM4E
SCHEMBL3963492 0.72 KDM4E (0.47) ALDH1A1ADORA3KDM4EHPGDTDP1
SCHEMBL3962364 0.72 IRAK4 (0.46) CLK4CYP1A2CYP3A4CYP2D6USP2
SCHEMBL18571767 0.72 PTGER4 (0.44) ALDH1A1HSD17B10ALOX15MEN1KMT2A
SCHEMBL5906640 0.71 F11 (0.47) GPR39CLK4CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034390-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C ARROW THERAPEUTICS LIMITED (GB) 2009-03-19 WO disclosed
WO-2009034390-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE IN TREATING HEPATITIS C ARROW THERAPEUTICS LIMITED (GB) 2009-03-19 WO disclosed