SCHEMBL3962971

SCHEMBL3962971

Nc1ccc(C(=O)NCCc2ccccc2)c(C(F)(F)F)n1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.52
RAB9A P51151 5/20 0.52
TAAR1 Q96RJ0 1/20 0.49
EGLN1 Q9GZT9 1/20 0.49
MLYCD O95822 2/20 0.49
HDAC4 P56524 2/20 0.47
GSK3B P49841 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3957622 0.80 RAB9A (0.58) NPC1RAB9AEGLN1MLYCDL3MBTL1
SCHEMBL28213665 0.75 NPC1 (0.56) NPC1RAB9AMLYCD
SCHEMBL13073725 0.74 NPC1 (0.66) NPC1RAB9AMLYCDHDAC4HDAC3
SCHEMBL1178776 0.74 HTT (0.59) NPC1RAB9ATAAR1MLYCDHDAC4
SCHEMBL29883463 0.73 GABRP (0.55) L3MBTL1
SCHEMBL5320191 0.72 NPC1 (0.67) NPC1RAB9AL3MBTL1HDAC6
SCHEMBL13541971 0.72 TAAR1 (0.54) NPC1RAB9ATAAR1MLYCDHDAC4
SCHEMBL27894530 0.71 NPC1 (0.56) NPC1RAB9AMLYCDHDAC4HDAC3
SCHEMBL3062674 0.70 MLYCD (0.76) NPC1RAB9ATAAR1MLYCDHDAC4
SCHEMBL16352053 0.69 RAB9A (0.62) NPC1RAB9AEGLN1L3MBTL1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079739-A2 PYRIDO[4,3-D]PYRIMIDIN-4(3H)-ONE DERIVATIVES AS CALCIUM RECEPTOR ANTAGONISTS Pfizer Products Inc. (US) 2009-07-22 EP disclosed
WO-2008041118-A2 PYRIDO[4,3-D]PYRIMIDIN-4(3H)-ONE DERIVATIVES AS CALCIUM RECEPTOR ANTAGONISTS PFIZER PRODUCTS INC. (US) 2008-04-10 WO disclosed