SCHEMBL3963549

SCHEMBL3963549

Cc1ccncc1C(=O)OCC(C)C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
TSHR P16473 1/20 0.56
TDP1 Q9NUW8 2/20 0.51
SIRT3 Q9NTG7 1/20 0.51
ADRB2 P07550 3/20 0.42
ADRB1 P08588 3/20 0.42
ADRB3 P13945 3/20 0.42
MAPT P10636 2/20 0.41
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
MEN1 O00255 1/20 0.40
TP53 P04637 1/20 0.40
NPY1R P25929 1/20 0.40
NPY2R P49146 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29570949 0.83 SIRT3 (0.58) ALDH1A1TSHRTDP1SIRT3NPC1
SCHEMBL907851 0.83 SIRT3 (0.58) ALDH1A1TSHRTDP1SIRT3NPC1
Ethane SCHEMBL28930003 0.82 SIRT3 (0.56) ALDH1A1TSHRTDP1SIRT3NPC1
SCHEMBL27349113 0.82 ALDH1A1 (0.57) ALDH1A1TSHRTDP1ADRB2ADRB1
SCHEMBL9260863 0.81 ALDH1A1 (0.56) ALDH1A1TSHRTDP1MAPTKDM4E
Iodomethane SCHEMBL10841815 0.81 SIRT3 (0.54) ALDH1A1TSHRTDP1SIRT3NPC1
SCHEMBL4591568 0.78 TDP1 (0.65) ALDH1A1TDP1SIRT3MAPTKDM4E
SCHEMBL27977119 0.77 TDP1 (0.50) ALDH1A1TSHRTDP1SIRT3MAPT
SCHEMBL27703244 0.77 L3MBTL1 (0.58) ALDH1A1TSHRTDP1SIRT3MAPT
SCHEMBL6057357 0.77 ALDH1A1 (0.79) ALDH1A1TSHRTDP1ADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-A2 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2009-07-22 EP disclosed
WO-2008038251-A2 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-04-03 WO disclosed