SCHEMBL3963722

SCHEMBL3963722

CN1CCN(Cc2ccc(C(=O)NN)c(C3CCCCC3)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.46
CSF1R P07333 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
FLT3 P36888 1/20 0.41
BTK Q06187 1/20 0.41
LMNA P02545 1/20 0.41
CHKA P35790 4/20 0.41
CHEK1 O14757 2/20 0.41
CA2 P00918 1/20 0.40
NCF1 P14598 1/20 0.40
PRMT6 Q96LA8 1/20 0.40
DDR1 Q08345 2/20 0.40
DDR2 Q16832 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
ALDH1A1 P00352 1/20 0.40
NUDT1 P36639 1/20 0.39
BACE1 P56817 1/20 0.39
ABL1 P00519 1/20 0.39
BCR P11274 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24728863 0.72 HDAC6 (0.78) HDAC6HRH3BTKLMNACHKA
SCHEMBL31721218 0.70 CHRM3 (0.61) HDAC6BTK
SCHEMBL9548868 0.69 ADRB3 (0.39) LMNAKDM4ENUDT1BACE1
SCHEMBL31553383 0.69 ALDH1A1 (0.48) HRH3KDM4EALDH1A1
SCHEMBL3954239 0.69 HDAC3 (0.52) LMNACA2KDM4EGAAALDH1A1
SCHEMBL27785362 0.69 HDAC6 (0.52) HDAC6HRH3BTKLMNACHKA
SCHEMBL16485458 0.69 CHKA (0.54) HDAC6CHKACHEK1KDM4E
Hydrochloric Acid SCHEMBL28314241 0.68 HDAC6 (0.51) HDAC6HRH3BTKLMNACHKA
SCHEMBL6188428 0.67 HDAC6 (0.54) HDAC6HRH3BTKLMNACHKA
SCHEMBL3953587 0.67 HDAC3 (0.50) LMNACA2KDM4EGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2077841-A1 NOVEL SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS Glaxo Group Limited (GB) 2009-07-15 EP disclosed
WO-2008052934-A1 NOVEL SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2008-05-08 WO disclosed