SCHEMBL3967588

SCHEMBL3967588

Clc1nc(-c2cc3ccccc3s2)c2cc[nH]c2n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGK1 P00558 1/20 0.38
APP P05067 2/20 0.37
DHPS P49366 1/20 0.37
PDK1 Q15118 1/20 0.37
PRKCQ Q04759 1/20 0.37
PRKCD Q05655 1/20 0.37
MAPKAPK2 P49137 1/20 0.36
NQO1 P15559 1/20 0.36
NQO2 P16083 1/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
CCNT1 O60563 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CDK9 P50750 1/20 0.35
IKBKB O14920 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3975335 0.83 CYP2A6 (0.38) PDK1ADORA2AADORA1CYP2A6
SCHEMBL28596883 0.75 CLK1 (0.47) APPDHPSPRKCQPRKCDMAPKAPK2
SCHEMBL30173282 0.75 CLK1 (0.47) APPDHPSPRKCQPRKCDMAPKAPK2
SCHEMBL3973616 0.74 ADORA2A (0.44) PDK1JAK2JAK3ADORA2AADORA1
SCHEMBL10125408 0.74 CCNK (0.44) PGK1APPDHPSPRKCQPRKCD
SCHEMBL13213033 0.73 JAK2 (0.56) PDK1PRKCQJAK2JAK3ADORA2A
SCHEMBL101422 0.71 CDK9 (0.54) PRKCQJAK2JAK3CCNT1CCNA2
SCHEMBL3971472 0.71 ADORA2A (0.38) PDK1PRKCQJAK2JAK3ADORA2A
SCHEMBL3975493 0.71 MEN1 (0.38) PDK1ADORA2AADORA1CYP2A6
SCHEMBL3975437 0.71 CDK1 (0.42) PRKCQPRKCDIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049028-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USE AS JANUS KINASE MODULATORS TARGEGEN INC. (US) 2009-04-16 WO disclosed
WO-2009049028-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USE AS JANUS KINASE MODULATORS TARGEGEN INC. (US) 2009-04-16 WO disclosed