SCHEMBL3971282

SCHEMBL3971282

N#Cc1ccc2cc(-c3nc(Nc4ccc(OCCC5CCCN5)cc4)nc4[nH]ccc34)sc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.36
CDK1 P06493 1/20 0.36
CCNB1 P14635 1/20 0.36
CDK2 P24941 1/20 0.36
CDK7 P50613 1/20 0.36
CDK9 P50750 1/20 0.36
CCNH P51946 1/20 0.36
CDK5 Q00535 1/20 0.36
JAK2 O60674 4/20 0.35
SLC6A4 P31645 2/20 0.35
JAK3 P52333 1/20 0.35
BTK Q06187 1/20 0.35
AURKB Q96GD4 1/20 0.34
TTBK1 Q5TCY1 1/20 0.34
TTBK2 Q6IQ55 1/20 0.34
CRBN Q96SW2 1/20 0.33
CTSS P25774 1/20 0.33
CHRNA1 P02708 1/20 0.33
CHRNG P07510 1/20 0.33
CHRNB1 P11230 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3969991 0.86 JAK3 (0.36) CCNT1CDK1CCNB1CDK2CDK7
SCHEMBL13883460 0.85 BACE1 (0.40) CDK1JAK2JAK3LTA4H
SCHEMBL3973959 0.81 JAK3 (0.38) CCNT1CDK1CCNB1CDK2CDK7
SCHEMBL3969959 0.81 JAK3 (0.38) CCNT1CDK1CCNB1CDK2CDK7
SCHEMBL3974063 0.80 JAK3 (0.40) CCNT1CDK1CCNB1CDK2CDK7
SCHEMBL3969296 0.79 BACE1 (0.40) CDK1JAK2JAK3LTA4H
SCHEMBL3974132 0.77 JAK3 (0.43) CCNT1CDK1CCNB1CDK2CDK7
SCHEMBL3976981 0.75 PRKCQ (0.44) CDK1CDK2CDK7CDK5JAK2
SCHEMBL3971424 0.74 TTK (0.56) JAK2JAK3BTK
SCHEMBL3966481 0.73 BACE1 (0.48) JAK2JAK3LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049028-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USE AS JANUS KINASE MODULATORS TARGEGEN INC. (US) 2009-04-16 WO disclosed