SCHEMBL4078130

SCHEMBL4078130

Nc1sc(-c2ccc(Cl)cc2)c(-c2cccc(C(F)(F)F)c2)c1-c1ccccc1C=O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.40
RORB Q92753 4/20 0.39
TP53 P04637 4/20 0.38
MDM2 Q00987 4/20 0.38
RORC P51449 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MAPT P10636 1/20 0.35
ADORA2A P29274 2/20 0.35
MAOB P27338 1/20 0.35
IDO1 P14902 1/20 0.34
IKBKB O14920 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4090647 0.93 ADORA1 (0.46) ADORA1RORBRORCNPC1RAB9A
SCHEMBL4076829 0.87 RORB (0.41) ADORA1RORBTP53RORCMAPT
SCHEMBL3974618 0.86 ADORA1 (0.44) ADORA1RORBRORCMAPTMAOB
SCHEMBL4080804 0.86 ADORA1 (0.43) ADORA1RORBRORCMAPTADORA2A
SCHEMBL3976889 0.82 ADORA1 (0.46) ADORA1RORBRORCMAPTMAOB
SCHEMBL4091364 0.82 ADORA1 (0.56) ADORA1RORBRORCMAPTADORA2A
SCHEMBL4078131 0.75 ADORA1 (0.68) ADORA1RORBTP53MDM2MAPT
SCHEMBL4085898 0.75 ADORA1 (0.42) ADORA1RORBRORCADORA2AMAOB
SCHEMBL2478195 0.73 RORC (0.50) ADORA1RORBRORCMAPTADORA2A
SCHEMBL3974628 0.70 GRM6 (0.61) ADORA1TP53MDM2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049362-A1 A1 ADENOSINE RECEPTOR ALLOSTERIC ENHANCERS MONASH UNIVERSITY (AU) 2009-04-23 WO disclosed