SCHEMBL3976889

SCHEMBL3976889

CC(=O)c1cccc(-c2sc(N)c(-c3ccccc3C=O)c2-c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.46
CNR2 P34972 2/20 0.40
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
RORB Q92753 5/20 0.37
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
MAOB P27338 2/20 0.36
LCK P06239 1/20 0.35
PTGS1 P23219 1/20 0.35
ERN1 O75460 1/20 0.35
RORC P51449 1/20 0.35
SLC9A1 P19634 1/20 0.35
HDAC2 Q92769 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3974618 0.93 ADORA1 (0.44) ADORA1CNR2ALDH1A1MEN1CYP1A2
SCHEMBL4090647 0.87 ADORA1 (0.46) ADORA1CNR2ALDH1A1RORBMAOB
SCHEMBL4078130 0.82 ADORA1 (0.40) ADORA1MAPTRORBMAOBRORC
SCHEMBL4076829 0.82 RORB (0.41) ADORA1ALDH1A1MEN1MAPTKMT2A
SCHEMBL3976892 0.80 ADORA1 (0.68) ADORA1CNR2ALDH1A1MEN1CYP1A2
SCHEMBL4091364 0.79 ADORA1 (0.56) ADORA1CNR2MAPTRORBMAOB
SCHEMBL4080804 0.79 ADORA1 (0.43) ADORA1CNR2MAPTRORBMAOB
SCHEMBL3981712 0.74 GRM6 (0.57) ADORA1ALDH1A1MEN1CYP1A2CYP3A4
SCHEMBL3974619 0.73 ADORA1 (0.67) ADORA1CNR2ALDH1A1MEN1CYP1A2
SCHEMBL4085898 0.72 ADORA1 (0.42) ADORA1CNR2ALDH1A1RORBMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049362-A1 A1 ADENOSINE RECEPTOR ALLOSTERIC ENHANCERS MONASH UNIVERSITY (AU) 2009-04-23 WO disclosed