SCHEMBL3974928

SCHEMBL3974928

CN(C)CCCc1c([N+](=O)[O-])cccc1S(N)(=O)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.47
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
TDP1 Q9NUW8 3/20 0.39
F2 P00734 2/20 0.39
PRSS1 P07477 2/20 0.39
PRSS2 P07478 2/20 0.39
PRSS3 P35030 2/20 0.39
BDKRB1 P46663 2/20 0.39
BDKRB2 P30411 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
DRD2 P14416 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
CHRM3 P20309 1/20 0.38
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7694792 0.79 F2 (0.47) ALDH1A1MEN1KMT2ACA2CA9
SCHEMBL30678498 0.78 F2 (0.45) ALDH1A1MEN1KMT2ACA2CA9
SCHEMBL1548597 0.75 FBP1 (0.45) ALDH1A1MEN1KMT2ACA2CA9
SCHEMBL1807309 0.74 TDP1 (0.62) SMN1; SMN2ALDH1A1MEN1KMT2ACA2
SCHEMBL28297463 0.73 HTR6 (0.42) CA2HTR2AHTR2CHTR2B
SCHEMBL6470839 0.73 MAPT (0.45) SMN1; SMN2ALDH1A1MEN1KMT2ACA2
SCHEMBL29052405 0.72 KMT2A (0.44) ALDH1A1MEN1KMT2ACA2CA9
SCHEMBL31437144 0.72 KMT2A (0.44) ALDH1A1MEN1KMT2ACA2CA9
SCHEMBL4690711 0.72 KMT2A (0.48) ALDH1A1MEN1KMT2ACA2CA9
SCHEMBL6468940 0.72 TDP1 (0.49) SMN1; SMN2ALDH1A1MEN1KMT2ACA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907385-A4 COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2009-05-06 EP disclosed
EP-1907385-A2 COMPOUNDS SmithKline Beecham Corporation (US) 2008-04-09 EP disclosed
WO-2007018941-A2 PYRIMIDYL-THIOPHENE DERIVATIVES SMITHKLINE BEECHAM CORPORATION (US) 2007-02-15 WO disclosed