SCHEMBL3975742

SCHEMBL3975742

O=C1CCC(C2CCCCC2)C1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.39
TRIM24 O15164 2/20 0.35
TRIM33 Q9UPN9 2/20 0.35
KMT2A Q03164 1/20 0.34
NOS1 P29475 3/20 0.31
NOS2 P35228 3/20 0.31
NOS3 P29474 2/20 0.31
MAP1LC3B Q9GZQ8 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
SLC18A3 Q16572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4864165 1.00 ALDH1A1 (0.40) ALDH1A1MAPTTRIM24TRIM33KMT2A
SCHEMBL28066099 0.97 ALDH1A1 (0.42) ALDH1A1MAPTTRIM24TRIM33KMT2A
SCHEMBL7009533 0.97 ALDH1A1 (0.42) ALDH1A1MAPTTRIM24TRIM33KMT2A
SCHEMBL1865812 0.97 ALDH1A1 (0.42) ALDH1A1MAPTTRIM24TRIM33KMT2A
SCHEMBL6889659 0.97 ALDH1A1 (0.42) ALDH1A1MAPTTRIM24TRIM33KMT2A
SCHEMBL6889662 0.97 ALDH1A1 (0.42) ALDH1A1MAPTTRIM24TRIM33KMT2A
SCHEMBL16512839 0.92 ALDH1A1 (0.35) ALDH1A1MAPTTRIM24TRIM33
SCHEMBL11593525 0.92 ALDH1A1 (0.35) ALDH1A1MAPTTRIM24TRIM33
SCHEMBL4866556 0.90 ALDH1A1 (0.41) ALDH1A1MAPTTRIM24TRIM33KMT2A
SCHEMBL11330899 0.90 TRIM24 (0.48) ALDH1A1MAPTTRIM24TRIM33KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874301-A4 NIACIN RECEPTOR AGONISTS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT MERCK & CO INC (US) 2009-05-06 EP disclosed
US-20090054423-A1 Niacin receptor agonists, compositions containing such compounds and methods of treatment MERCK SHARP & DOHME CORP. 2009-02-26 US disclosed
US-20080125310-A1 Hydride reduction of alpha, beta-unsaturated carbonyl compounds using chiral organic catalysts CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2008-05-29 US disclosed
US-7323604-B2 Hydride reduction of α,β-unsaturated carbonyl compounds using chiral organic catalysts CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2008-01-29 US disclosed
EP-1874301-A1 NIACIN RECEPTOR AGONISTS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT Merck & Co., Inc. (US) 2008-01-09 EP disclosed
WO-2006113150-A1 NIACIN RECEPTOR AGONISTS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT MERCK & CO., INC. (US) 2006-10-26 WO disclosed
US-20060161024-A1 Hydride reduction of alpha, beta-unsaturated carbonyl compounds using chiral organic catalysts CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2006-07-20 US disclosed
US-4251398-A FOR ENHANCING OTHER ODORS, SCENTING TOILETRIES FIRMENICH SA (CH) 1981-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054423-A1 Niacin receptor agonists, compositions containing such compounds and methods of treatment FFAR1, HCAR1, GPR119 ALDH1A1 949/4885MAPT 2698/4885TRIM24 4294/4885
US-20060161024-A1 Hydride reduction of alpha, beta-unsaturated carbonyl compounds using chiral organic catalysts ECH1, CBR1, DHCR24 ALDH1A1 14/4885MAPT 2535/4885TRIM24 1676/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.