SCHEMBL3978066

SCHEMBL3978066

CCN1CCCC(Cc2cccnc2)C1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.50
CHRNA4 P43681 2/20 0.50
CHRM2 P08172 2/20 0.50
CHRM1 P11229 2/20 0.50
CHRM3 P20309 2/20 0.50
CARM1 Q86X55 1/20 0.49
PRMT6 Q96LA8 1/20 0.49
HRH3 Q9Y5N1 1/20 0.47
CHRNA7 P36544 3/20 0.47
GBA1 P04062 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
KDM4E B2RXH2 1/20 0.44
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12090436 0.85 CHRM2 (0.64) CHRNB2CHRNA4CHRM2CHRM1CHRM3
SCHEMBL3979979 0.83 CARM1 (0.50) CARM1PRMT6HRH3
SCHEMBL9912161 0.83 PRMT6 (0.68) CARM1PRMT6
SCHEMBL12424313 0.81 CHRNB2 (0.61) CHRNB2CHRNA4CHRM2CHRM1CHRM3
SCHEMBL12255644 0.80 CHRM2 (0.49) CHRNB2CHRNA4CHRM2CHRM1CHRM3
SCHEMBL20268602 0.79 ALDH1A1 (0.54) CHRNB2CHRNA4CHRM2CHRM1CHRM3
SCHEMBL2743291 0.79 CHRM2 (0.68) CHRNB2CHRNA4CHRM2CHRM1CHRM3
SCHEMBL31054426 0.77 CHRNA7 (0.53) CHRNB2CHRNA4CHRM2CHRM1CHRM3
SCHEMBL27686945 0.77 KDM4E (0.56) CHRNB2CHRNA4CHRM2CHRM1CHRM3
SCHEMBL9534698 0.77 CHRNA7 (0.53) CHRNB2CHRNA4CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009056693-A1 NOVEL DERIVATIVES OF N, N'- 2, 4-DIANILINOPYRIMIDINES, PREPARATION THEREOF AS MEDICAMENTS PHARMACEUTICAL COMPOSITIONS AND IN PARTICULAR AS IKK INHIBITORS SANOFI-AVENTIS (FR) 2009-05-07 WO disclosed