SCHEMBL3978601

SCHEMBL3978601

Nc1ccc(N2C(=O)CN(N3CC(=O)N(c4ccc([N+](=O)[O-])cc4)C3=O)C2=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
SCN2A Q99250 1/20 0.45
MAPT P10636 5/20 0.45
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
PKM P14618 2/20 0.42
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
CTSG P08311 1/20 0.42
CMA1 P23946 1/20 0.42
ESR1 P03372 1/20 0.40
CYP19A1 P11511 1/20 0.40
ESR2 Q92731 1/20 0.40
POLB P06746 2/20 0.40
APEX1 P27695 1/20 0.40
CASP6 P55212 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
SIRT6 Q8N6T7 2/20 0.39
ADRB1 P08588 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL854476 0.77 SIRT6 (0.49) ALDH1A1SCN2AMAPTKMT2AMEN1
SCHEMBL3978598 0.77 ALDH1A1 (0.53) ALDH1A1SCN2AMAPTKMT2AMEN1
SCHEMBL10643664 0.76 SCN2A (0.54) ALDH1A1SCN2AMAPTKMT2AMEN1
SCHEMBL5314298 0.76 ENPP2 (0.41) ALDH1A1SCN2AMAPTPOLB
4-Nitroaniline SCHEMBL16451 0.73 ALDH1A1 (1.00) ALDH1A1MAPTKMT2AMEN1PKM
4-Nitroaniline SCHEMBL27963818 0.73 ALDH1A1 (1.00) ALDH1A1MAPTKMT2AMEN1PKM
SCHEMBL9065915 0.73 ALDH1A1 (1.00) ALDH1A1MAPTKMT2AMEN1PKM
4-Nitroaniline SCHEMBL13529022 0.73 ALDH1A1 (1.00) ALDH1A1MAPTKMT2AMEN1PKM
SCHEMBL2557016 0.72 SCN2A (0.58) ALDH1A1SCN2AMAPTKMT2AMEN1
4-Nitroaniline SCHEMBL29077543 0.71 ALDH1A1 (0.86) ALDH1A1MAPTKMT2AMEN1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907385-A4 COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2009-05-06 EP disclosed
EP-1907385-A2 COMPOUNDS SmithKline Beecham Corporation (US) 2008-04-09 EP disclosed
WO-2007018941-A2 PYRIMIDYL-THIOPHENE DERIVATIVES SMITHKLINE BEECHAM CORPORATION (US) 2007-02-15 WO disclosed