SCHEMBL3979300

SCHEMBL3979300

Cc1cccc2c1c(C(=O)c1cc(Cl)ncn1)cn2C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 1/20 0.36
CMA1 P23946 8/20 0.35
CTSG P08311 1/20 0.35
POLB P06746 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
LCK P06239 1/20 0.34
RORC P51449 2/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
MAOB P27338 1/20 0.33
MITF O75030 1/20 0.33
ALDH1A1 P00352 1/20 0.33
USP2 O75604 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3988367 0.87 RORC (0.40) POLBKMT2AMEN1RORCMAOB
SCHEMBL3989803 0.85 ABCG2 (0.39) KMT2AMEN1RAB9ARORCMAPT
SCHEMBL4257168 0.83 POLB (0.33) CDK2POLBKMT2ALMNAMAPT
SCHEMBL4259652 0.82 NR4A2 (0.34) CDK2KMT2AMEN1NPC1RAB9A
SCHEMBL3972624 0.81 POLB (0.55) POLBKMT2AMEN1NPC1RAB9A
SCHEMBL3990181 0.81 RORC (0.39) CDK2POLBKMT2AMEN1RORC
SCHEMBL3992240 0.78 POLB (0.38) CDK2POLBKMT2ALMNAMAPT
SCHEMBL3996013 0.78 KDR (0.41) CDK2POLBKMT2AMEN1LMNA
SCHEMBL3995880 0.76 NTRK1 (0.33)
SCHEMBL3992947 0.76 POLB (0.38) CDK2POLBKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2065382-A1 CGRP antagonists Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2009-06-03 EP disclosed
WO-2009050235-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed