SCHEMBL3988367

SCHEMBL3988367

Cn1cc(C(=O)c2cc(Cl)ncn2)c2c(F)cccc21

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RORC P51449 6/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2C9 P11712 3/20 0.40
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.38
CNR1 P21554 4/20 0.37
CNR2 P34972 1/20 0.37
CHRM1 P11229 2/20 0.36
POLB P06746 1/20 0.36
CYP2C19 P33261 1/20 0.35
NTRK1 P04629 2/20 0.35
PCSK9 Q8NBP7 1/20 0.35
SCN9A Q15858 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3979300 0.87 CDK2 (0.36) RORCCYP2C9MEN1ALDH1A1KMT2A
SCHEMBL3995880 0.85 NTRK1 (0.33) NTRK1PCSK9
SCHEMBL3989803 0.84 ABCG2 (0.39) RORCMEN1ALDH1A1KMT2ACNR2
SCHEMBL4257168 0.82 POLB (0.33) ALDH1A1KMT2APOLBCYP2C19MAOB
SCHEMBL3994459 0.81 PCSK9 (0.51) RORCCYP3A4CYP2C9CNR1CNR2
SCHEMBL4259652 0.81 NR4A2 (0.34) RORCMEN1ALDH1A1KMT2ACYP2C19
SCHEMBL3972624 0.81 POLB (0.55) MEN1ALDH1A1KMT2APOLBMAOB
SCHEMBL1742839 0.79 CES2 (0.46) ALDH1A1
SCHEMBL3973248 0.78 KDM4E (0.42) RORCALDH1A1CNR1CNR2POLB
SCHEMBL3978572 0.78 PCSK9 (0.40) RORCMEN1ALDH1A1KMT2ACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2065382-A1 CGRP antagonists Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2009-06-03 EP disclosed