SCHEMBL3983196

SCHEMBL3983196

NNC(=O)c1c(C(=O)OC(=O)c2occ(-c3ccccc3)c2-c2ccccc2)ccc(O)c1F

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 1/20 0.32
HSD17B2 P37059 1/20 0.32
ALOX15 P16050 1/20 0.32
ALOX12 P18054 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TLR9 Q9NR96 1/20 0.32
KAT6A Q92794 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3981614 0.91 ALOX15 (0.34) ALOX15ALOX12ALDH1A1MAPTMEN1
SCHEMBL3982435 0.90 ALOX15 (0.38) ALOX15ALOX12MAPTMEN1KMT2A
SCHEMBL3981082 0.89 MEN1 (0.34) ALOX15ALOX12ALDH1A1MAPTMEN1
SCHEMBL3982135 0.89 MEN1 (0.34) ALOX15ALOX12ALDH1A1MAPTL3MBTL1
SCHEMBL3973512 0.88 ALOX15 (0.32) ALOX15ALOX12GAA
SCHEMBL3983965 0.88 ALOX15 (0.32) ALOX15ALOX12ALDH1A1MAPTGAA
SCHEMBL3978772 0.87 TACR1 (0.31) ALOX15ALOX12ALDH1A1
SCHEMBL3982340 0.87 CTSD (0.36) ALDH1A1MAPT
SCHEMBL3977753 0.86 PDE4B (0.35) ALDH1A1MAPTMEN1KMT2AGAA
SCHEMBL3975937 0.85 ALDH1A1 (0.36) ALOX15ALOX12ALDH1A1MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7514452-B2 2-furancarboxylic acid hydrazides and pharmaceutical compositions containing the same DAINIPPON PHARMACEUTICAL CO., LTD (JP) 2009-04-07 US disclosed
US-20050171196-A1 2-Furancarboxylic acid hydrazides and pharmaceutical compositions containing the same DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2005-08-04 US disclosed
EP-1489077-A1 2-FURANCARBOXYLIC ACID HYDRAZIDES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2004-12-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050171196-A1 2-Furancarboxylic acid hydrazides and pharmaceutical compositions containing the same GLP1R, GCGR, GPR119 HSD17B1 919/4885HSD17B2 832/4885ALOX15 2249/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.