SCHEMBL3984777

SCHEMBL3984777

CCC1CN(c2nc3c(C(=O)O)cccc3o2)CCN1Cc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 6/20 0.40
HTR6 P50406 6/20 0.39
NAAA Q02083 4/20 0.39
KCNH2 Q12809 2/20 0.39
HCAR2 Q8TDS4 1/20 0.39
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA9 Q16790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1004886 0.81 HTR3A (0.46) HTR3AHTR6CA1CA2CA4
SCHEMBL1004885 0.81 HTR3A (0.46) HTR3AHTR6CA1CA2CA4
SCHEMBL3987869 0.76 NAAA (0.39) HTR3AHTR6NAAAKCNH2HCAR2
SCHEMBL1004342 0.74 HTR6 (0.58) HTR3AHTR6NAAAKCNH2HCAR2
SCHEMBL3990768 0.74 HTR3A (0.50) HTR3AKCNH2
SCHEMBL1005851 0.74 HTR3A (0.50) HTR3AKCNH2
SCHEMBL1006017 0.74 HTR3A (0.66) HTR3AKCNH2
SCHEMBL1004971 0.74 HTR3A (0.66) HTR3AKCNH2
SCHEMBL1004970 0.74 HTR3A (0.66) HTR3AKCNH2
SCHEMBL1004188 0.73 HTR3A (0.48) HTR3AHTR6LMNACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed