SCHEMBL3987336

SCHEMBL3987336

COC(=O)c1cccc2oc(N3CC(C)NC(C)C3)nc12

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 13/20 0.48
TOP2A P11388 2/20 0.47
KCNH2 Q12809 3/20 0.44
HCRTR1 O43613 3/20 0.42
HCRTR2 O43614 3/20 0.42
CYP2C19 P33261 1/20 0.41
FGFR1 P11362 1/20 0.41
RIPK1 Q13546 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1005033 0.87 HTR3A (0.61) HTR3ATOP2AKCNH2HCRTR1HCRTR2
SCHEMBL3990476 0.87 HTR3A (0.61) HTR3ATOP2AKCNH2HCRTR1HCRTR2
SCHEMBL3990473 0.87 HTR3A (0.61) HTR3ATOP2AKCNH2HCRTR1HCRTR2
SCHEMBL1006005 0.81 TOP2A (0.50) HTR3ATOP2AKCNH2RIPK1
SCHEMBL1007867 0.81 ALDH1A1 (0.48) HTR3ATOP2AKCNH2
SCHEMBL1007229 0.80 HTR6 (0.52) HTR3ATOP2AKCNH2
SCHEMBL1004911 0.80 HTR3A (0.59) HTR3ATOP2AKCNH2CYP2C19
SCHEMBL1007287 0.80 HTR3A (0.48) HTR3ATOP2AKCNH2RIPK1
SCHEMBL1004565 0.80 HTR3A (0.61) HTR3ATOP2AKCNH2CYP2C19RIPK1
SCHEMBL3984677 0.80 HTR3A (0.61) HTR3ATOP2AKCNH2CYP2C19RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed