SCHEMBL3987977

SCHEMBL3987977

NC(=O)N1CCC2(CC1)NCNC2=O

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.40
HTT P42858 1/20 0.40
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PARP1 P09874 1/20 0.35
CRBN Q96SW2 3/20 0.34
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
CDK19 Q9BWU1 1/20 0.33
DDB1 Q16531 2/20 0.33
KCNH2 Q12809 1/20 0.32
HDAC1 Q13547 1/20 0.32
FPR2 P25090 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3989054 0.84 CRBN (0.38) PARP1CRBNCCNCCDK8CDK19
SCHEMBL14414389 0.80 ALDH1A1 (0.44) HTTKDM4EALDH1A1PARP1CRBN
SCHEMBL18347987 0.79 CHRNB2 (0.38) PARP1CRBNCCNCCDK8CDK19
SCHEMBL20215842 0.79 OPRM1 (0.39) ALDH1A1PARP1CRBNCCNCCDK8
SCHEMBL29889238 0.74 CRBN (0.59) GAAHTTKDM4EALDH1A1CRBN
SCHEMBL21634313 0.72 ALDH1A1 (0.48) GAAALDH1A1CRBNDDB1
SCHEMBL31622202 0.71 GAA (0.40) GAAHTTKDM4EALDH1A1CRBN
SCHEMBL5562592 0.70 HIF1A (0.56) ALDH1A1
SCHEMBL9963246 0.70 CYP2D6 (0.36) GAAKDM4EALDH1A1CCNCCDK8
SCHEMBL29890275 0.70 OTUD7B (0.46) GAAHTTKDM4EALDH1A1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035420-A2 KV1.5 POTASSIUM CHANNEL INHIBITORS Wyeth a Corporation of the State of Delaware (US) 2009-03-18 EP claimed
WO-2007149873-A2 KV1.5 POTASSIUM CHANNEL INHIBITORS WYETH (US) 2007-12-27 WO claimed