SCHEMBL3973248

SCHEMBL3973248

Cn1cc(C(=O)c2cc(Cl)ncn2)c2cc(F)ccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
RORC P51449 1/20 0.38
PCSK9 Q8NBP7 1/20 0.38
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
POLB P06746 1/20 0.36
KCNH2 Q12809 2/20 0.36
GSK3B P49841 2/20 0.36
CDK2 P24941 1/20 0.36
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
NR4A2 P43354 3/20 0.36
MAPK14 Q16539 2/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
AURKA O14965 1/20 0.34
JAK2 O60674 1/20 0.34
PAK4 O96013 1/20 0.34
ABL1 P00519 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3978572 0.91 PCSK9 (0.40) KDM4EALDH1A1RORCPCSK9CNR1
SCHEMBL3996013 0.88 KDR (0.41) KDM4EALDH1A1CNR1CNR2POLB
SCHEMBL3972624 0.84 POLB (0.55) ALDH1A1POLBNR4A2
SCHEMBL3986985 0.84 ABCG2 (0.47) KDM4EALDH1A1GSK3BNR4A2JAK2
SCHEMBL3992240 0.81 POLB (0.38) ALDH1A1CNR1CNR2POLBCDK2
SCHEMBL3992947 0.81 POLB (0.38) KDM4EALDH1A1CNR1CNR2POLB
SCHEMBL3989840 0.80 MTNR1A (0.39) CA12CA9NR4A2
SCHEMBL3995936 0.79 ALDH1A1 (0.44) ALDH1A1CNR2POLBKDM4CROCK1
SCHEMBL3995880 0.79 NTRK1 (0.33) PCSK9KCNH2CA12CA9MAPK14
SCHEMBL3997478 0.79 POLB (0.36) KDM4EALDH1A1CNR1CNR2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2065382-A1 CGRP antagonists Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2009-06-03 EP disclosed
WO-2009050235-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed