SCHEMBL3989034

SCHEMBL3989034

CC(C)C(C(=O)N(C)C(CO)Cc1ccc(O)c(C(C)(C)C)c1)N(C)CC(N)Cc1ccc(F)cc1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.33
OPRD1 P41143 4/20 0.32
OPRK1 P41145 4/20 0.32
OPRM1 P35372 1/20 0.30
REN P00797 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3987590 0.90 MAOB (0.33) TRPA1OPRD1OPRK1REN
SCHEMBL3986378 0.88 FCER2 (0.30) REN
SCHEMBL3995150 0.83 CYP3A4 (0.35) TRPA1OPRD1OPRM1REN
SCHEMBL3989091 0.82 REN (0.34) OPRD1OPRK1OPRM1REN
SCHEMBL3987434 0.81 ALOX15 (0.32) TRPA1OPRD1OPRK1OPRM1
SCHEMBL3989149 0.81 BACE1 (0.36) OPRD1OPRK1REN
SCHEMBL3990161 0.79 F2R (0.30)
SCHEMBL3993021 0.75 TRPA1 (0.33) TRPA1
SCHEMBL3994857 0.75 ACACB (0.33) OPRD1OPRK1OPRM1REN
SCHEMBL13795944 0.75 SLC7A5 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553969-B1 Substituted phenethylamine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-06-30 US disclosed
EP-1149843-A1 SUBSTITUTED PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-10-31 EP disclosed