SCHEMBL3989149

SCHEMBL3989149

CC(C)C(C(=O)NC(CN)Cc1ccc(O)c(C(C)(C)C)c1)N(C)CC(N)Cc1ccc(F)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.36
AKT1 P31749 2/20 0.34
AKT2 P31751 2/20 0.34
AKT3 Q9Y243 2/20 0.34
REN P00797 1/20 0.33
CIT O14578 1/20 0.32
ROCK2 O75116 1/20 0.32
PRKCB P05771 1/20 0.32
PRKCA P17252 1/20 0.32
PRKACA P17612 1/20 0.32
PRKACB P22694 1/20 0.32
ROCK1 Q13464 1/20 0.32
PKN1 Q16512 1/20 0.32
PRKD2 Q9BZL6 1/20 0.32
FCER2 P06734 1/20 0.32
MC4R P32245 1/20 0.32
MC3R P41968 1/20 0.32
OPRK1 P41145 5/20 0.32
MME P08473 2/20 0.32
ACE P12821 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3995150 0.94 CYP3A4 (0.35) BACE1RENFCER2MC4RMC3R
SCHEMBL3989091 0.91 REN (0.34) RENROCK2ROCK1FCER2OPRK1
SCHEMBL3987590 0.83 MAOB (0.33) RENOPRK1OPRD1
SCHEMBL3994857 0.82 ACACB (0.33) RENROCK2ROCK1FCER2OPRK1
SCHEMBL3989034 0.81 TRPA1 (0.33) RENOPRK1OPRD1
SCHEMBL3986378 0.81 FCER2 (0.30) RENFCER2
SCHEMBL13796438 0.80 MC4R (0.37) BACE1RENMC4RMC3RMME
SCHEMBL13796434 0.79 MC4R (0.36) BACE1RENFCER2MC4RMC3R
SCHEMBL3989491 0.77 MC4R (0.35) RENFCER2MC4RMC3ROPRK1
SCHEMBL3989661 0.77 BACE1 (0.34) BACE1RENMC4RMC3RBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553969-B1 Substituted phenethylamine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-06-30 US disclosed
EP-1149843-A1 SUBSTITUTED PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-10-31 EP disclosed