SCHEMBL3989527

SCHEMBL3989527

Cc1cc(=O)nc(C(N)Cc2ccc(O)c(C(C)(C)C)c2)[nH]1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 11/20 0.34
ALOX15 P16050 5/20 0.34
HSD17B10 Q99714 4/20 0.34
KDM4E B2RXH2 3/20 0.34
RECQL P46063 3/20 0.34
HIF1A Q16665 3/20 0.34
USP2 O75604 2/20 0.34
ADORA3 P0DMS8 2/20 0.34
HTR2A P28223 2/20 0.34
PTGS2 P35354 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
EGFR P00533 1/20 0.34
LCK P06239 1/20 0.34
FYN P06241 1/20 0.34
PTGS1 P23219 1/20 0.34
SLC7A5 Q01650 1/20 0.34
ROCK1 Q13464 3/20 0.33
ALDH1A1 P00352 3/20 0.33
SCN10A Q9Y5Y9 2/20 0.33
NR1I2 O75469 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3989532 0.84 HSD17B10 (0.36) ROCK2ALOX15HSD17B10KDM4ERECQL
SCHEMBL3988348 0.77 PTPRB (0.32) ALOX15HSD17B10KDM4ERECQLHIF1A
SCHEMBL3994642 0.70 TAAR1 (0.52) ALOX15HSD17B10KDM4ERECQLHIF1A
SCHEMBL18194421 0.69 ALOX15 (0.51) ALOX15HSD17B10KDM4ERECQLHIF1A
SCHEMBL14856009 0.68 SLC7A5 (0.67) ALOX15HSD17B10KDM4ERECQLHIF1A
SCHEMBL10656842 0.68 SLC7A5 (0.67) ALOX15HSD17B10KDM4ERECQLHIF1A
SCHEMBL7892985 0.68 SLC7A5 (0.67) ALOX15HSD17B10KDM4ERECQLHIF1A
SCHEMBL3985975 0.68 ALDH1A1 (0.43) ALOX15HSD17B10KDM4ERECQLHIF1A
SCHEMBL3985972 0.68 ALOX15 (0.43) ALOX15HSD17B10KDM4ERECQLHIF1A
SCHEMBL29809967 0.68 SLC7A5 (0.67) ALOX15HSD17B10KDM4ERECQLHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553969-B1 Substituted phenethylamine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-06-30 US disclosed
EP-1149843-A1 SUBSTITUTED PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-10-31 EP disclosed