SCHEMBL3989532

SCHEMBL3989532

Cc1cc(=O)[nH]c(C(N)Cc2ccc(O)c(C(C)(C)C)c2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.36
KDM4E B2RXH2 1/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 1/20 0.36
GAA P10253 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
POLB P06746 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
ROCK2 O75116 3/20 0.34
ALDH1A1 P00352 2/20 0.33
SCN10A Q9Y5Y9 2/20 0.33
LMNA P02545 2/20 0.33
HTT P42858 2/20 0.33
NR1I2 O75469 1/20 0.33
CYP2C9 P11712 1/20 0.33
MIF P14174 1/20 0.33
TYR P14679 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3989527 0.84 ROCK2 (0.34) HSD17B10KDM4EHPGDMAPK1POLB
SCHEMBL3988353 0.77 MMP13 (0.36) KDM4EMAPK1GAAHDAC6POLB
SCHEMBL3994642 0.70 TAAR1 (0.52) HSD17B10KDM4EHPGDMAPK1POLB
SCHEMBL18194421 0.69 ALOX15 (0.51) HSD17B10KDM4EHPGDMAPK1GAA
SCHEMBL10656842 0.68 SLC7A5 (0.67) HSD17B10KDM4EHPGDPOLBHSP90AA1
SCHEMBL7892985 0.68 SLC7A5 (0.67) HSD17B10KDM4EHPGDPOLBHSP90AA1
SCHEMBL14856009 0.68 SLC7A5 (0.67) HSD17B10KDM4EHPGDPOLBHSP90AA1
SCHEMBL3985975 0.68 ALDH1A1 (0.43) HSD17B10KDM4EHPGDMAPK1GAA
SCHEMBL3985970 0.68 ALOX15 (0.43) HSD17B10KDM4EHPGDMAPK1GAA
SCHEMBL29809967 0.68 SLC7A5 (0.67) HSD17B10KDM4EHPGDPOLBHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553969-B1 Substituted phenethylamine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-06-30 US disclosed
EP-1149843-A1 SUBSTITUTED PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-10-31 EP disclosed