SCHEMBL3988348

SCHEMBL3988348

CNC(C(=O)NC(Cc1ccc(O)c(C(C)(C)C)c1)c1nc(=O)cc(C)[nH]1)C(C)C

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRB P23467 1/20 0.32
MRE11 P49959 2/20 0.31
SCN10A Q9Y5Y9 1/20 0.30
ALOX15 P16050 3/20 0.30
ALOX12 P18054 3/20 0.30
KDM4E B2RXH2 2/20 0.30
MEN1 O00255 2/20 0.30
ALDH1A1 P00352 2/20 0.30
ESR1 P03372 2/20 0.30
TP53 P04637 2/20 0.30
CYP3A4 P08684 2/20 0.30
HPGD P15428 2/20 0.30
MAPK1 P28482 2/20 0.30
RECQL P46063 2/20 0.30
KMT2A Q03164 2/20 0.30
HIF1A Q16665 2/20 0.30
HSD17B10 Q99714 2/20 0.30
NR1I2 O75469 1/20 0.30
GMNN O75496 1/20 0.30
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3988353 0.88 MMP13 (0.36) PTPRBSCN10AKDM4EMAPK1LMNA
SCHEMBL3993261 0.84 PSMB11 (0.34) CYP3A4NR1I2NR3C1CYP1A2CYP2D6
SCHEMBL3987600 0.78
SCHEMBL4657375 0.77 ACACB (0.38) ALOX15ALOX12KDM4EMEN1ALDH1A1
SCHEMBL3989527 0.77 ROCK2 (0.34) SCN10AALOX15ALOX12KDM4EMEN1
SCHEMBL3987548 0.75 ERCC1 (0.30)
SCHEMBL3986499 0.75 PTPRB (0.40) PTPRBMRE11ALOX15ALOX12TP53
SCHEMBL3994576 0.73 ROCK2 (0.30)
SCHEMBL3993264 0.72 MAPT (0.36) CYP3A4NR1I2NR3C1CYP1A2POLB
SCHEMBL3988356 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553969-B1 Substituted phenethylamine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-06-30 US disclosed
EP-1149843-A1 SUBSTITUTED PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-10-31 EP disclosed