SCHEMBL3996320

SCHEMBL3996320

CC(C)(C)OC(=O)N1CCC(n2c(CNC3CCCc4cccnc43)nc3ccccc32)CC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 4/20 0.52
OPRM1 P35372 5/20 0.46
OGFRL1 Q5TC84 5/20 0.46
OPRD1 P41143 4/20 0.46
NOD2 Q9HC29 1/20 0.44
NOD1 Q9Y239 1/20 0.44
OPRK1 P41145 3/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
KDM1A O60341 1/20 0.42
CCR5 P51681 3/20 0.41
FNTA P49354 2/20 0.41
FNTB P49356 2/20 0.41
RORC P51449 1/20 0.40
GPR119 Q8TDV5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3999603 0.88 CXCR4 (0.53) CXCR4OPRM1OGFRL1OPRD1OPRK1
SCHEMBL3373812 0.86 CXCR4 (0.56) CXCR4NOD2NOD1HDAC1HDAC6
SCHEMBL4939959 0.84 CXCR4 (0.74) CXCR4OPRM1OGFRL1OPRD1NOD2
SCHEMBL4885774 0.80 CXCR4 (0.47) CXCR4HDAC1HDAC6KDM1AFNTA
SCHEMBL4885422 0.79 CXCR4 (0.49) CXCR4HDAC1HDAC6KDM1AFNTA
Trifluoroacetic Acid SCHEMBL4889301 0.77 CXCR4 (0.44) CXCR4HDAC1HDAC6KDM1AFNTA
SCHEMBL4716688 0.76 HDAC1 (0.52) CXCR4HDAC1HDAC6
SCHEMBL18661189 0.76 CXCR4 (0.49) CXCR4OPRM1OGFRL1OPRD1OPRK1
SCHEMBL2084608 0.76 FNTA (0.51) CXCR4HDAC1HDAC6KDM1AFNTA
SCHEMBL14130832 0.76 LMNA (0.57) CXCR4HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778231-A4 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2009-06-03 EP disclosed
US-20080096861-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION (US) 2008-04-24 US disclosed
EP-1778231-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-02 EP disclosed
WO-2006020415-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080096861-A1 Chemical Compounds CCR5, CXCR4, CXCR3 CXCR4 2/4885OPRM1 257/4885OGFRL1 264/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.