Clobetasol Propionate

Clobetasol Propionate

SCHEMBL3997

CCC(=O)O[C@]1(C(=O)CCl)[C@@H](C)C[C@H]2[C@@H]3CCC4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@@]21C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1

The experimentally established mechanism targets of Clobetasol Propionate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 6/20 1.00
PGR P06401 6/20 1.00
CYP3A4 P08684 5/20 1.00
USP2 O75604 5/20 1.00
LMNA P02545 3/20 1.00
MAPT P10636 3/20 1.00
NR1I2 O75469 2/20 1.00
SMN1; SMN2 Q16637 2/20 1.00
NPSR1 Q6W5P4 2/20 1.00
MLNR O43193 1/20 1.00
ABCB11 O95342 1/20 1.00
CYP3A5 P20815 1/20 1.00
PPARG P37231 1/20 1.00
CYP2D6 P10635 1/20 1.00
CYP2C9 P11712 1/20 1.00
ADORA3 P0DMS8 3/20 0.84
DRD2 P14416 1/20 0.84
OPRD1 P41143 1/20 0.84
MEN1 O00255 1/20 0.75
KMT2A Q03164 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Clobetasol Propionate SCHEMBL5577907 1.00 PGR (1.00) PGRNR3C1CYP3A4USP2LMNA
Clobetasol Propionate SCHEMBL17131797 1.00 PGR (1.00) PGRNR3C1CYP3A4USP2LMNA
Clobetasol Propionate SCHEMBL11052078 1.00 PGR (1.00) PGRNR3C1CYP3A4USP2LMNA
Clobetasol Propionate SCHEMBL11052079 1.00 PGR (1.00) PGRNR3C1CYP3A4USP2LMNA
Clobetasol Propionate SCHEMBL445257 1.00 PGR (1.00) PGRNR3C1CYP3A4USP2LMNA
Clobetasol Propionate SCHEMBL5577908 1.00 PGR (1.00) PGRNR3C1CYP3A4USP2LMNA
Clobetasol Propionate SCHEMBL10865006 1.00 PGR (1.00) PGRNR3C1CYP3A4USP2LMNA
Clobetasol Propionate SCHEMBL28118983 0.98 NR3C1 (0.95) PGRNR3C1CYP3A4USP2LMNA
Betamethasone Dipropionate SCHEMBL18301225 0.95 NR3C1 (0.93) PGRNR3C1CYP3A4USP2LMNA
SCHEMBL596943 0.94 NR3C1 (0.88) PGRNR3C1CYP3A4USP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 34992 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137656-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
US-20260137657-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
US-20260139030-A1 CHIMERIC PROTEINS FOR TREATING CUTANEOUS INFLAMMATION SHATTUCK LABS INC (US) 2026-05-21 US claimed
EP-4744657-A1 THERAPEUTIC AGENT FOR HUMAN GRAFT VERSUS HOST DISEASE AND COMBINATION THEREOF National University Corporation Okayama University (JP) 2026-05-20 EP claimed
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
US-20260130899-A1 METHOD OF TREATMENT FOR PREVENTION OF GLUCOCORTICOID TOXICITY AND/OR ENHANCEMENT OF MUSCLE REGENERATION VIA NEUTROPHIL ELASTASE INHIBITION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2026-05-14 US claimed
EP-4741421-A1 FAB-ARM EXCHANGE-PREVENTING FC VARIANTS FROM WHICH EFFECTOR FUNCTIONS ARE REMOVED Korea University Research and Business Foundation (KR) 2026-05-13 EP claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-3222270-B1 COMPOSITIONS FOR MUCOSAL ADHESION AND USES THEREOF BIONANOPLUS S L (ES) 2026-04-29 EP claimed
US-20260103492-A1 CYCLOSPORINE COMPOSITIONS AND METHODS OF USE BACAINN BIOTHERAPEUTICS, LTD. (KY) 2026-04-16 US claimed
EP-0216453-A2 Esters of hyaluronic acid and their salts. FIDIA S.p.A. (IT) 1987-04-01 EP claimed
EP-0197718-A2 New medicaments for topical use FIDIA S.p.A. (IT) 1986-10-15 EP claimed
EP-0173478-A1 Treatment of skin disorders SCOTIA HOLDINGS PLC (GB) 1986-03-05 EP claimed
EP-0068553-B1 TOPICAL ANTIMICROBIAL ANTI-INFLAMMATORY COMPOSITIONS THE PROCTER & GAMBLE COMPANY (US) 1985-11-21 EP claimed
US-4370322-A BETAMETHASONE, BECLOMETHASONE AND CLOBETASOL DERIVATIVES GLAXO GROUP LIMITED (GB) 1983-01-25 US claimed
EP-0068553-A1 Topical antimicrobial anti-inflammatory compositions THE PROCTER & GAMBLE COMPANY (US) 1983-01-05 EP claimed
US-4343798-A Topical antimicrobial anti-inflammatory compositions THE PROCTER & GAMBLE COMPANY (US) 1982-08-10 US claimed
US-4333927-A CORTICOSTEROID, PHOSPHATIDE, BUTYLHYDROXYANISOLE AND/OR BUTYLHYDROXYTOLUENE MITSUBISHI CHEMICAL INDUSTRIES, LTD. (JP) 1982-06-08 US claimed
US-4244942-A Creamy preparation containing steroid and process for the preparation thereof TOKO YAKUHIN KOGYO KABUSHIKI KAISHA (JP) 1981-01-13 US claimed
US-4083974-A Topical steroidal anti-inflammatory preparations containing polyoxypropylene 15 stearyl ether THE UPJOHN COMPANY (US) 1978-04-11 US claimed