SCHEMBL4002037

SCHEMBL4002037

Cc1cc(Cl)cnc1CCCC(=O)N1CCc2c(Cl)c(O)c(O)c(Cl)c2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.39
RAB9A P51151 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
KMT2A Q03164 1/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAPK1 P28482 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SMYD3 Q9H7B4 1/20 0.35
PTGDR2 Q9Y5Y4 4/20 0.34
HTR5A P47898 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13963199 0.92 HPGD (0.39) HPGDRAB9ANPSR1MEN1NPC1
SCHEMBL4006857 0.89 HPGD (0.41) HPGDRAB9ANPSR1MEN1NPC1
SCHEMBL4016104 0.88 AGBL2 (0.41) HPGDNPSR1MEN1KMT2AMAPT
SCHEMBL13963197 0.84 TRPV1 (0.34) HPGDNPSR1MAPTALDH1A1TSHR
SCHEMBL4009380 0.80 HPGD (0.39) HPGDRAB9ANPSR1MEN1KMT2A
SCHEMBL4011125 0.80 ALDH1A1 (0.37) NPSR1MEN1KMT2AMAPTALDH1A1
SCHEMBL13962555 0.79 MAPT (0.43) RAB9ANPSR1MEN1NPC1KMT2A
SCHEMBL13962550 0.79 MAPT (0.37) RAB9ANPSR1MEN1NPC1KMT2A
SCHEMBL4010973 0.77 ENPP2 (0.41) HPGDRAB9AMAPTTSHRMAPK1
SCHEMBL13963201 0.77 PTGDR2 (0.42) HPGDTSHRTAAR1SMN1; SMN2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007418-A1 NOVEL BRONCHODILATING ISOQUINOLINE AMIDES RESPIRATORIUS AB (SE) 2009-01-15 WO disclosed
WO-2009007418-A1 NOVEL BRONCHODILATING ISOQUINOLINE AMIDES RESPIRATORIUS AB (SE) 2009-01-15 WO disclosed