SCHEMBL4002268

SCHEMBL4002268

CC(C)(C)OC(=O)Cn1cc(-c2ccccc2Cl)c2c(C#N)ncnc21

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 5/20 0.36
CNR2 P34972 5/20 0.36
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
BTK Q06187 4/20 0.34
PIK3CD O00329 1/20 0.33
CFD P00746 1/20 0.33
BCL6 P41182 1/20 0.33
P2RX7 Q99572 2/20 0.33
KLKB1 P03952 1/20 0.32
FPR2 P25090 1/20 0.32
EIF2AK3 Q9NZJ5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13769690 0.85 STAT3 (0.38) PIK3CDCFDBCL6KLKB1
SCHEMBL4012260 0.79 FPR2 (0.33) KDM4EALDH1A1KLKB1FPR2
SCHEMBL4009501 0.79 SCN9A (0.36) CNR1CNR2KDM4EALDH1A1P2RX7
SCHEMBL13769756 0.75 VEGFA (0.37) ALDH1A1EIF2AK3
SCHEMBL19208112 0.75 CFD (0.37) KDM4EALDH1A1CFDBCL6P2RX7
SCHEMBL13769532 0.74 PDE4B (0.41) KDM4EALDH1A1P2RX7
SCHEMBL19208282 0.73 HDAC6 (0.39) KDM4EALDH1A1FPR2
SCHEMBL4006140 0.72 CNR1 (0.56) CNR1CNR2KDM4EALDH1A1
SCHEMBL13769525 0.72 MAPT (0.40) CNR1CNR2KDM4EALDH1A1P2RX7
SCHEMBL13769936 0.71 PDE4B (0.42) KDM4EALDH1A1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed