SCHEMBL4009501

SCHEMBL4009501

CC(C)(C)OC(=O)Cn1cc(-c2cccc(Cl)c2Cl)c2c(Cl)ncnc21

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.36
CCR4 P51679 6/20 0.35
FPR2 P25090 1/20 0.35
EIF2AK3 Q9NZJ5 1/20 0.34
CNR1 P21554 3/20 0.34
CNR2 P34972 3/20 0.34
P2RX7 Q99572 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 2/20 0.33
SRC P12931 1/20 0.32
MEN1 O00255 1/20 0.32
NR2F2 P24468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4008416 0.84 CCR4 (0.39) CCR4EIF2AK3CNR2P2RX7KMT2A
SCHEMBL4002268 0.79 CNR1 (0.36) FPR2EIF2AK3CNR1CNR2P2RX7
SCHEMBL13769680 0.79 MAPK14 (0.40) CCR4EIF2AK3P2RX7KDM4EALDH1A1
SCHEMBL4007105 0.78 ADK (0.40) FPR2P2RX7KDM4EALDH1A1KMT2A
SCHEMBL13769532 0.78 PDE4B (0.41) P2RX7KDM4EALDH1A1KMT2ASRC
SCHEMBL4012559 0.76 CCR4 (0.40) CCR4EIF2AK3P2RX7SRC
SCHEMBL19208112 0.75 CFD (0.37) FPR2P2RX7KDM4EALDH1A1KMT2A
SCHEMBL4007615 0.74 SRC (0.43) CCR4P2RX7KMT2ASRCMEN1
SCHEMBL4013000 0.74 CCR4 (0.39) CCR4P2RX7
SCHEMBL25542303 0.74 FPR2 (0.33) FPR2KDM4EALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed