SCHEMBL4007932

SCHEMBL4007932

O[C@@H]1[C@@H](OCc2ccccc2)[C@@H](O)O[C@H](COCc2ccccc2)[C@H]1OCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GJB2 P29033 4/20 0.53
TACR2 P21452 3/20 0.50
HTR1A P08908 1/20 0.47
NT5E P21589 1/20 0.47
GJA1 P17302 2/20 0.46
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
PDE4D Q08499 1/20 0.43
SLC6A2 P23975 1/20 0.43
SSTR1 P30872 1/20 0.43
SSTR2 P30874 1/20 0.43
SSTR4 P31391 1/20 0.43
SSTR3 P32745 1/20 0.43
SSTR5 P35346 1/20 0.43
PTPN1 P18031 2/20 0.42
CDC25B P30305 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4007928 1.00 GJB2 (0.53) GJB2TACR2HTR1ANT5EGJA1
SCHEMBL21843054 1.00 GJB2 (0.53) GJB2TACR2HTR1ANT5EGJA1
SCHEMBL7150778 1.00 GJB2 (0.53) GJB2TACR2HTR1ANT5EGJA1
SCHEMBL7150775 1.00 GJB2 (0.53) GJB2TACR2HTR1ANT5EGJA1
SCHEMBL13797895 1.00 GJB2 (0.53) GJB2TACR2HTR1ANT5EGJA1
SCHEMBL5473075 0.93 GJB2 (0.52) GJB2TACR2HTR1ANT5EGJA1
SCHEMBL9114888 0.93 GJB2 (0.47) GJB2TACR2HTR1ANT5EBCHE
SCHEMBL13430417 0.93 GJB2 (0.52) GJB2TACR2HTR1ANT5EGJA1
SCHEMBL9114883 0.93 GJB2 (0.47) GJB2TACR2HTR1ANT5EBCHE
SCHEMBL13430414 0.93 GJB2 (0.52) GJB2TACR2HTR1ANT5EGJA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7541456-B2 Enolization; dimerization; trimerization; for synthesis of sugar molecules CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2009-06-02 US disclosed
EP-1501777-A4 DIRECT, ENANTIOSELECTIVE ALDOL COUPLING OF ALDEHYDES USING CHIRAL ORGANIC CATALYSTS CALIFORNIA INST OF TECHN (US) 2007-03-28 EP disclosed
US-20050197498-A1 Enolization; dimerization; trimerization; for synthesis of sugar molecules CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2005-09-08 US disclosed
US-6900357-B2 Comprises (2S,5S)-5-benzyl-2-tert-butyl-3-methylimidazolidin-4-one as catalyst; for synthesis of (2S,3S)-3-hydroxy-2-methylpentanal CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2005-05-31 US disclosed
EP-1501777-A1 DIRECT, ENANTIOSELECTIVE ALDOL COUPLING OF ALDEHYDES USING CHIRAL ORGANIC CATALYSTS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2005-02-02 EP disclosed
US-20040024221-A1 Comprises (2S,5S)-5-benzyl-2-tert-butyl-3-methylimidazolidin-4-one as catalyst; for synthesis of (2S,3S)-3-hydroxy-2-methylpentanal MACMILLAN DAVID W C (US) 2004-02-05 US disclosed
WO-2003089396-A1 DIRECT, ENANTIOSELECTIVE ALDOL COUPLING OF ALDEHYDES USING CHIRAL ORGANIC CATALYSTS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2003-10-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040024221-A1 Comprises (2S,5S)-5-benzyl-2-tert-butyl-3-methylimidazolidin-4-one as catalyst; for synthesis of (2S,3S)-3-hydroxy-2-methylpentanal ADH1C, ADH5, ALDH3A1 GJB2 2098/4885TACR2 3744/4885HTR1A 1947/4885
US-20050197498-A1 Enolization; dimerization; trimerization; for synthesis of sugar molecules DERA, ALDOA, TALDO1 GJB2 1333/4885TACR2 2297/4885HTR1A 3292/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.