SCHEMBL4010033

SCHEMBL4010033

O=CCCc1ccc(C(F)(F)F)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 3/20 0.50
TRPV4 Q9HBA0 1/20 0.44
TKT P29401 1/20 0.39
KDM1A O60341 2/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
KCNH2 Q12809 2/20 0.36
HTR2A P28223 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
NAMPT P43490 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP3A5 P20815 1/20 0.34
PPARD Q03181 1/20 0.34
PLAAT3 P53816 1/20 0.34
PLAAT5 Q96KN8 1/20 0.34
PLAAT2 Q9NWW9 1/20 0.34
PLAAT4 Q9UL19 1/20 0.34
KCNQ3 O43525 1/20 0.34
KCNQ2 O43526 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL934661 0.84 TRPV4 (0.48) DAOTRPV4TKTKDM1AMAOA
Hydrochloric Acid SCHEMBL4727675 0.81 TRPV4 (0.46) DAOTRPV4TKTKDM1AMAOA
SCHEMBL13680809 0.78 GRIN1 (0.41) MRGPRX4GRIN1GRIN2B
SCHEMBL3842669 0.78 KDM1A (0.47) DAOTRPV4KDM1AMAOAMAOB
SCHEMBL22558739 0.78 L3MBTL1 (0.50) KCNH2TRPV1
SCHEMBL264730 0.77 TAAR1 (0.52) DAOTRPV4TKTKDM1AMAOA
SCHEMBL694114 0.77 DAO (0.50) DAOTRPV4TKTKDM1AMAOA
SCHEMBL19615786 0.77 TRPV4 (0.53) DAOTRPV4TKTKDM1AMAOA
SCHEMBL3851699 0.77 DAO (0.50) DAOTRPV4TKTKDM1AMAOA
SCHEMBL1259004 0.77 TKT (0.55) DAOTRPV4TKTKDM1AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009085256-A1 ANTI-HIV COMPOUNDS PANACOS PHARMACEUTICALS, INC. (US) 2009-07-09 WO disclosed
WO-2009085256-A1 ANTI-HIV COMPOUNDS PANACOS PHARMACEUTICALS, INC. (US) 2009-07-09 WO disclosed