SCHEMBL4010343

SCHEMBL4010343

[CH2]Oc1ccc(C(N)c2ccc(OC)cc2OC)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
ALDH1A1 P00352 5/20 0.42
CYP3A4 P08684 1/20 0.42
ADRA2A P08913 2/20 0.42
ADRA1A P35348 2/20 0.42
CYP2D6 P10635 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPK1 P28482 1/20 0.41
BLM P54132 1/20 0.41
BCHE P06276 1/20 0.40
TYR P14679 1/20 0.40
ACHE P22303 1/20 0.40
HTR2A P28223 1/20 0.40
CYP1A1 P04798 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4010346 0.90 CA12 (0.48) CA12CA1CA2CA7CA9
SCHEMBL6386316 0.84 BCHE (0.50) CA12CA1CA2CA7CA9
SCHEMBL3140878 0.84 CA1 (0.43) CA12CA1CA2CA7CA9
SCHEMBL414370 0.84 MEN1 (0.48) CA12CA1CA2CA7CA9
SCHEMBL2632344 0.83 BCHE (0.46) CA12CA1CA2CA7CA9
SCHEMBL11399910 0.83 CA12 (0.56) CA12CA1CA2CA7CA9
SCHEMBL16437139 0.82 CA12 (0.41) CA12CA1CA2CA7CA9
SCHEMBL7145569 0.81 LMNA (0.46) CA12CA1CA2CA7CA9
SCHEMBL16351174 0.80 SLC2A1 (0.46) CA12CA1CA2CA7CA9
SCHEMBL17189617 0.80 HTR2A (0.42) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1713493-A4 PITUITARY ADENYLATE CYCLASE ACTIVATING PEPTIDE (PACAP) RECEPTOR (VPAC2) AGONISTS AND THEIR PHARMACOLOGICAL METHODS OF USE BAYER PHARMACEUTICALS CORP (US) 2009-06-24 EP disclosed
US-20090143283-A1 Pituitary Adenylate Cyclase Activating Peptide (PACAP) Receptor (VPAC2) Agonists and Their Pharmacological Methods of Use BAYER PHARMACEUTICALS CORPORATION (US) 2009-06-04 US disclosed
EP-1713493-A2 PITUITARY ADENYLATE CYCLASE ACTIVATING PEPTIDE (PACAP) RECEPTOR (VPAC2) AGONISTS AND THEIR PHARMACOLOGICAL METHODS OF USE Bayer Pharmaceuticals Corporation (US) 2006-10-25 EP disclosed
WO-2005072385-A2 PITUITARY ADENYLATE CYCLASE ACTIVATING PEPTIDE (PACAP) RECEPTOR (VPAC2) AGONISTS AND THEIR PHARMACOLOGICAL METHODS OF USE BAYER PHARMACEUTICALS CORPORATION (US) 2005-08-11 WO disclosed