SCHEMBL4258452

SCHEMBL4258452

Cc1cc(C(N)=O)c(NCC(C)CC(F)(F)F)cc1C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM6B O15054 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
CASR P41180 1/20 0.32
MAPK14 Q16539 1/20 0.31
HSP90AA1 P07900 4/20 0.31
HSP90AB1 P08238 4/20 0.31
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
TAS2R14 Q9NYV8 2/20 0.30
NNMT P40261 1/20 0.30
CISD1 Q9NZ45 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2428070 0.83 MEN1 (0.47) MEN1TSHRKMT2AKDM6BKDM4C
SCHEMBL3973224 0.82 CISD1 (0.36) MEN1TSHRKMT2AKDM6BKDM4C
SCHEMBL2425954 0.82 HSP90AA1 (0.39) CASRMAPK14HSP90AA1HSP90AB1RXRA
SCHEMBL3979062 0.81 CISD1 (0.38) MEN1TSHRKMT2AKDM6BKDM4C
SCHEMBL2434508 0.80 CISD1 (0.34) MAPK14HSP90AA1HSP90AB1RXRARXRB
SCHEMBL3975210 0.79 CASR (0.33) MEN1TSHRKMT2AKDM6BKDM4C
SCHEMBL3975516 0.78 RXRB (0.34) KDM4CMAPK14HSP90AA1HSP90AB1RXRA
SCHEMBL4010874 0.78 GUCY1A1 (0.40) KDM6BKDM4CHSP90AA1HSP90AB1NNMT
SCHEMBL2422460 0.75 JAK2 (0.40) HSP90AA1HSP90AB1NNMTCISD1
SCHEMBL2424120 0.73 JAK2 (0.34) HSP90AA1HSP90AB1RXRARXRBTAS2R14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed