SCHEMBL4012181

SCHEMBL4012181

CS(=O)(=O)c1cccc2c(-c3cc(O)ccc3Cl)ccnc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.45
NR1H2 P55055 5/20 0.43
NR1H3 Q13133 5/20 0.43
COMT P21964 4/20 0.40
PDE4D Q08499 3/20 0.39
MMP14 P50281 2/20 0.37
PIK3CD O00329 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
MEN1 O00255 2/20 0.37
HSP90AA1 P07900 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALOX15B O15296 1/20 0.37
NR1I2 O75469 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
CYP3A4 P08684 1/20 0.37
HTR1A P08908 1/20 0.37
ALOX5 P09917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4299566 0.85 NR1H2 (0.50) PTGDR2NR1H2NR1H3COMTPIK3CD
SCHEMBL4011482 0.83 NR1H2 (0.47) PTGDR2NR1H2NR1H3PDE4DMEN1
SCHEMBL4011946 0.82 NR4A2 (0.49) PTGDR2NR1H2NR1H3PDE4DMMP14
SCHEMBL4018063 0.81 NR1H2 (0.55) PTGDR2NR1H2NR1H3SLC40A1RXRA
SCHEMBL4018184 0.81 PIK3CD (0.54) PTGDR2NR1H2NR1H3PIK3CDRXRA
SCHEMBL17044063 0.80 KDR (0.46) PTGDR2COMTMEN1HSP90AA1KMT2A
SCHEMBL4011996 0.79 NR1H2 (0.66) PTGDR2NR1H2NR1H3RXRA
SCHEMBL4012347 0.79 NR1H3 (0.45) PTGDR2NR1H2NR1H3PDE4DHTR1A
SCHEMBL4012339 0.78 NR1H2 (0.49) PTGDR2NR1H2NR1H3PDE4DMEN1
SCHEMBL17044086 0.78 RIPK2 (0.43) PTGDR2COMTMEN1HSP90AA1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed