SCHEMBL4012347

SCHEMBL4012347

CS(=O)(=O)c1cccc2c(-c3cc(OS(=O)(=O)C(F)(F)F)ccc3Cl)ccnc12

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 10/20 0.45
NR1H2 P55055 9/20 0.45
RXRA P19793 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.40
PDE4A P27815 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
CHRM1 P11229 5/20 0.35
DRD2 P14416 4/20 0.35
DRD4 P21917 4/20 0.35
DRD3 P35462 4/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
HTR2C P28335 1/20 0.34
HTR7 P34969 1/20 0.34
HTR6 P50406 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016970 0.88 NR1H3 (0.50) NR1H3NR1H2RXRAPTGDR2PDE4A
SCHEMBL4012080 0.88 NR1H2 (0.47) NR1H3NR1H2RXRAPTGDR2PDE4A
SCHEMBL4011482 0.86 NR1H2 (0.47) NR1H3NR1H2RXRAPTGDR2PDE4A
SCHEMBL4013386 0.85 PTGDR2 (0.39) NR1H3NR1H2RXRAPTGDR2PDE4A
SCHEMBL4011996 0.81 NR1H2 (0.66) NR1H3NR1H2RXRAPTGDR2
SCHEMBL4017522 0.80 NR1H2 (0.45) NR1H3NR1H2RXRAPTGDR2PDE4A
SCHEMBL4018729 0.79 NR1H2 (0.53) NR1H3NR1H2RXRAPTGDR2
SCHEMBL4012181 0.79 PTGDR2 (0.45) NR1H3NR1H2RXRAPTGDR2PDE4D
SCHEMBL4012339 0.78 NR1H2 (0.49) NR1H3NR1H2RXRAPTGDR2PDE4A
SCHEMBL4012778 0.78 NR1H2 (0.56) NR1H3NR1H2RXRAPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed